4XNV
The human P2Y1 receptor in complex with BPTU
Summary for 4XNV
Entry DOI | 10.2210/pdb4xnv/pdb |
Related | 4XNW |
Descriptor | P2Y purinoceptor 1, Rubredoxin, P2Y purinoceptor 1, 1-[2-(2-tert-butylphenoxy)pyridin-3-yl]-3-[4-(trifluoromethoxy)phenyl]urea, CHOLESTEROL, ... (8 entities in total) |
Functional Keywords | human p2y1 receptor, g protein coupled receptor, platelet activation, membrane protein, inhibitor complex, transport protein-inhibitor complex, psi-biology, structural genomics, gpcr network, gpcr, transport protein/inhibitor |
Biological source | Homo sapiens (Human) More |
Total number of polymer chains | 1 |
Total formula weight | 52916.56 |
Authors | Zhang, D.,Gao, Z.,Jacobson, K.,Han, G.W.,Stevens, R.,Zhao, Q.,Wu, B.,GPCR Network (GPCR) (deposition date: 2015-01-16, release date: 2015-04-01, Last modification date: 2020-02-05) |
Primary citation | Zhang, D.,Gao, Z.G.,Zhang, K.,Kiselev, E.,Crane, S.,Wang, J.,Paoletta, S.,Yi, C.,Ma, L.,Zhang, W.,Han, G.W.,Liu, H.,Cherezov, V.,Katritch, V.,Jiang, H.,Stevens, R.C.,Jacobson, K.A.,Zhao, Q.,Wu, B. Two disparate ligand-binding sites in the human P2Y1 receptor Nature, 520:317-321, 2015 Cited by PubMed: 25822790DOI: 10.1038/nature14287 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.2 Å) |
Structure validation
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