4R6A
Crystal structure of human TLR8 in complex with Hybrid-2
4R6A の概要
エントリーDOI | 10.2210/pdb4r6a/pdb |
分子名称 | Toll-like receptor 8, alpha-D-mannopyranose-(1-3)-beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... (7 entities in total) |
機能のキーワード | rna recognition, ssrna, leucine rich repeat, rna receptor, innate immunity, glycosylation, secreted, structure-based ligand design, vaccine adjuvants, antiviral and antitumor drug binding, rna binding protein |
由来する生物種 | Homo sapiens (human) |
タンパク質・核酸の鎖数 | 2 |
化学式量合計 | 192351.16 |
構造登録者 | |
主引用文献 | Ganapathi, L.,Haren, S.V.,Dowling, D.J.,Bergelson, I.,Shukla, N.M.,Malladi, S.S.,Balakrishna, R.,Tanji, H.,Ohto, U.,Shimizu, T.,David, S.A.,Levy, O. Hybrid-2: AnImidazoquinoline Dual Toll-like receptor 7/8 Agonist that Potently Activates Cytokine Production by Human Newborn and Adult Leukocytes To be Published, |
実験手法 | X-RAY DIFFRACTION (2.1 Å) |
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