4P44
X-ray structure of human glutamate carboxypeptidase II (GCPII) in complex with a phosphoramidate inhibitor JRB-4-81
4P44 の概要
エントリーDOI | 10.2210/pdb4p44/pdb |
分子名称 | Glutamate carboxypeptidase 2, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, alpha-D-mannopyranose-(1-3)-beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... (9 entities in total) |
機能のキーワード | prostate-specific membrane antigen, naaladase, phosphoramidate, hydrolase |
由来する生物種 | Homo sapiens (Human) |
細胞内の位置 | Cell membrane ; Single-pass type II membrane protein . Isoform PSMA': Cytoplasm : Q04609 |
タンパク質・核酸の鎖数 | 1 |
化学式量合計 | 83056.05 |
構造登録者 | |
主引用文献 | Novakova, Z.,Cerny, J.,Choy, C.J.,Nedrow, J.R.,Choi, J.K.,Lubkowski, J.,Berkman, C.E.,Barinka, C. Design of composite inhibitors targeting glutamate carboxypeptidase II: the importance of effector functionalities. Febs J., 283:130-143, 2016 Cited by PubMed: 26460595DOI: 10.1111/febs.13557 主引用文献が同じPDBエントリー |
実験手法 | X-RAY DIFFRACTION (1.75 Å) |
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