4NR8
Crystal structure of the first bromodomain of human BRD4 in complex with an isoxazolyl-benzimidazole ligand
4NR8 の概要
エントリーDOI | 10.2210/pdb4nr8/pdb |
分子名称 | Bromodomain-containing protein 4, POTASSIUM ION, 5-(3,5-dimethyl-1,2-oxazol-4-yl)-1-[2-(morpholin-4-yl)ethyl]-2-(2-phenylethyl)-1H-benzimidazole, ... (5 entities in total) |
機能のキーワード | structural genomics consortium, sgc, chemical tool, small molecule inhibitor, transcription, transcription-inhibitor complex, transcription/inhibitor |
由来する生物種 | Homo sapiens (human) |
細胞内の位置 | Nucleus: O60885 |
タンパク質・核酸の鎖数 | 1 |
化学式量合計 | 15631.09 |
構造登録者 | Filippakopoulos, P.,Picaud, S.,Felletar, I.,Hay, D.,Fedorov, O.,Martin, S.,von Delft, F.,Brennan, P.,Arrowsmith, C.H.,Edwards, A.M.,Bountra, C.,Knapp, S.,Structural Genomics Consortium (SGC) (登録日: 2013-11-26, 公開日: 2013-12-25, 最終更新日: 2023-09-20) |
主引用文献 | Filippakopoulos, P.,Hay, D.,von Delft, F.,Edwards, A.M.,Picaud, S.,Fedorov, O.,Brennan, P.,Bountra, C. Crystal structure of the first bromodomain of human BRD4 in complex with an isoxazolyl-benzimidazole ligand To be Published, |
実験手法 | X-RAY DIFFRACTION (1.635 Å) |
構造検証レポート
検証レポート(詳細版)をダウンロード