4KA2
Crystal structure of CD4-mimetic miniprotein M48U12 in complex with HIV-1 YU2 gp120
Summary for 4KA2
Entry DOI | 10.2210/pdb4ka2/pdb |
Related | 2I5Y 2I60 4JZW 4JZZ 4K0A |
Related PRD ID | PRD_001102 |
Descriptor | HIV-1 YU2 gp120, M48U12, 2-acetamido-2-deoxy-beta-D-glucopyranose, ... (4 entities in total) |
Functional Keywords | viral protein-peptide complex, hiv-1, gp120, yu2, cd4 mimic, m48u12, viral protein-inhibitor complex, viral protein/inhibitor |
Biological source | Human immunodeficiency virus 1 More |
Total number of polymer chains | 2 |
Total formula weight | 46520.89 |
Authors | Acharya, P.,Kwong, P.D. (deposition date: 2013-04-21, release date: 2013-06-19, Last modification date: 2023-11-15) |
Primary citation | Morellato-Castillo, L.,Acharya, P.,Combes, O.,Michiels, J.,Descours, A.,Ramos, O.H.,Yang, Y.,Vanham, G.,Arien, K.K.,Kwong, P.D.,Martin, L.,Kessler, P. Interfacial Cavity Filling To Optimize CD4-Mimetic Miniprotein Interactions with HIV-1 Surface Glycoprotein. J.Med.Chem., 56:5033-5047, 2013 Cited by PubMed: 23710622DOI: 10.1021/jm4002988 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.79 Å) |
Structure validation
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