4J4N
Crystal structure of FK506 binding domain of plasmodium falciparum FKBP35 in complex with D44
Summary for 4J4N
Entry DOI | 10.2210/pdb4j4n/pdb |
Related | 2OFN 2VN1 4J4O |
Descriptor | FK506-binding protein (FKBP)-type peptidyl-propyl isomerase, N-(2-ethylphenyl)-2-(3H-imidazo[4,5-b]pyridin-2-ylsulfanyl)acetamide (3 entities in total) |
Functional Keywords | d44, fkbp35, fk506 binding, isomerase-isomerase inhibitor complex, isomerase/isomerase inhibitor |
Biological source | Plasmodium falciparum |
Total number of polymer chains | 3 |
Total formula weight | 44531.43 |
Authors | Sreekanth, R.,Harikishore, A.,Yoon, H.S. (deposition date: 2013-02-07, release date: 2013-09-11, Last modification date: 2024-10-09) |
Primary citation | Harikishore, A.,Niang, M.,Rajan, S.,Preiser, P.R.,Yoon, H.S. Small molecule Plasmodium FKBP35 inhibitor as a potential antimalaria agent. Sci Rep, 3:2501-2501, 2013 Cited by PubMed: 23974147DOI: 10.1038/srep02501 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.75 Å) |
Structure validation
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