4F9Y
Human P38 alpha MAPK In Complex With a Novel and Selective Small Molecule Inhibitor
4F9Y の概要
エントリーDOI | 10.2210/pdb4f9y/pdb |
関連するPDBエントリー | 4EWQ 4F9W 4FA2 |
分子名称 | Mitogen-activated protein kinase 14, 4-[3-(4-FLUOROPHENYL)-1H-PYRAZOL-4-YL]PYRIDINE, N,N-dimethyl-6-(naphthalen-1-yl)-5-(pyridin-4-yl)pyridazin-3-amine, ... (6 entities in total) |
機能のキーワード | protein kinase catalytic domain, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
由来する生物種 | Homo sapiens (human) |
タンパク質・核酸の鎖数 | 1 |
化学式量合計 | 45023.18 |
構造登録者 | Grum-Tokars, V.L.,Minasov, G.,Anderson, W.F.,Watterson, D.M. (登録日: 2012-05-21, 公開日: 2013-06-05, 最終更新日: 2020-01-01) |
主引用文献 | Watterson, D.M.,Grum-Tokars, V.L.,Roy, S.M.,Schavocky, J.P.,Bradaric, B.D.,Bachstetter, A.D.,Xing, B.,Dimayuga, E.,Saeed, F.,Zhang, H.,Staniszewski, A.,Pelletier, J.C.,Minasov, G.,Anderson, W.F.,Arancio, O.,Van Eldik, L.J. Development of Novel In Vivo Chemical Probes to Address CNS Protein Kinase Involvement in Synaptic Dysfunction. Plos One, 8:e66226-e66226, 2013 Cited by PubMed: 23840427DOI: 10.1371/journal.pone.0066226 主引用文献が同じPDBエントリー |
実験手法 | X-RAY DIFFRACTION (1.85 Å) |
構造検証レポート
検証レポート(詳細版)をダウンロード