4BBM
CRYSTAL STRUCTURE OF THE HUMAN CDKL2 KINASE DOMAIN WITH BOUND TCS 2312
Summary for 4BBM
Entry DOI | 10.2210/pdb4bbm/pdb |
Related | 4AAA |
Descriptor | CYCLIN-DEPENDENT KINASE-LIKE 2, 4'-[5-[[3-[(CYCLOPROPYLAMINO)METHYL]PHENYL]AMINO]-1H-PYRAZOL-3-YL]-[1,1'-BIPHENYL]-2,4-DIOL, CHLORIDE ION, ... (5 entities in total) |
Functional Keywords | transferase, phospho-mimetic |
Biological source | HOMO SAPIENS (HUMAN) |
Cellular location | Cytoplasm : Q92772 |
Total number of polymer chains | 2 |
Total formula weight | 77925.06 |
Authors | Canning, P.,Elkins, J.M.,Cooper, C.D.O.,Mahajan, P.,Daga, N.,Berridge, G.,Burgess-Brown, N.,Muniz, J.R.C.,Krojer, T.,Arrowsmith, C.H.,Edwards, A.M.,Bountra, C.,von Delft, F.,Bullock, A. (deposition date: 2012-09-26, release date: 2012-10-17, Last modification date: 2023-12-20) |
Primary citation | Canning, P.,Park, K.,Goncalves, J.,Li, C.,Howard, C.J.,Sharpe, T.D.,Holt, L.J.,Pelletier, L.,Bullock, A.N.,Leroux, M.R. CDKL Family Kinases Have Evolved Distinct Structural Features and Ciliary Function. Cell Rep, 22:885-894, 2018 Cited by PubMed: 29420175DOI: 10.1016/j.celrep.2017.12.083 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2 Å) |
Structure validation
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