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4TKY

The complex structure of E. coli DsbA bound to a peptide at the DsbA/DsbB interface

Summary for 4TKY
Entry DOI10.2210/pdb4tky/pdb
DescriptorThiol:disulfide interchange protein DsbA, PRO-PHE-ALA-THR-CYS-ASP-SER, ACETYL GROUP, ... (5 entities in total)
Functional Keywordsdsba, dsbb, dithiol oxidase, complex, dsba/dsbb, peptide inhibitor, thioredoxin-related protein, oxidoreductase-peptide inhibitor complex, oxidoreductase/peptide inhibitor
Biological sourceEscherichia coli
More
Total number of polymer chains8
Total formula weight88496.04
Authors
Premkumar, L.,Martin, J.L. (deposition date: 2014-05-28, release date: 2015-01-14, Last modification date: 2023-09-27)
Primary citationDuprez, W.,Premkumar, L.,Halili, M.A.,Lindahl, F.,Reid, R.C.,Fairlie, D.P.,Martin, J.L.
Peptide Inhibitors of the Escherichia coli DsbA Oxidative Machinery Essential for Bacterial Virulence.
J.Med.Chem., 58:577-587, 2015
Cited by
PubMed: 25470204
DOI: 10.1021/jm500955s
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.5 Å)
Structure validation

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