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3WJ5

Crystal structure of PPARgamma ligand binding domain in complex with triphenyltin

Summary for 3WJ5
Entry DOI10.2210/pdb3wj5/pdb
Related3WJ4
DescriptorPeroxisome proliferator-activated receptor gamma, triphenylstannanyl (3 entities in total)
Functional Keywordsprotein-ligand complex, dna-binding, metal-binding, nucleus, receptor, transcription
Biological sourceHomo sapiens (human)
Total number of polymer chains2
Total formula weight63516.98
Authors
Harada, S.,Hiromori, Y.,Fukakusa, S.,Kawahara, K.,Nakamura, S.,Noda, M.,Uchiyama, S.,Fukui, K.,Nishikawa, J.,Nagase, H.,Kobayashi, Y.,Ohkubo, T.,Yoshida, T.,Nakanishi, T. (deposition date: 2013-10-04, release date: 2014-10-15, Last modification date: 2024-03-20)
Primary citationHarada, S.,Hiromori, Y.,Fukakusa, S.,Kawahara, K.,Nakamura, S.,Noda, M.,Uchiyama, S.,Fukui, K.,Nishikawa, J.,Nagase, H.,Kobayashi, Y.,Ohkubo, T.,Yoshida, T.,Nakanishi, T.
Structural basis for PPARgamma transactivation by endocrine disrupting organotin compounds
To be Published,
Experimental method
X-RAY DIFFRACTION (1.89 Å)
Structure validation

218853

数据于2024-04-24公开中

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