3VN2
Crystal Structure of PPARgamma complexed with Telmisartan
Summary for 3VN2
Entry DOI | 10.2210/pdb3vn2/pdb |
Descriptor | Peroxisome proliferator-activated receptor gamma, Nuclear receptor coactivator 1, 4'-[(1,7'-dimethyl-2'-propyl-1H,3'H-2,5'-bibenzimidazol-3'-yl)methyl]biphenyl-2-carboxylic acid, ... (4 entities in total) |
Functional Keywords | signaling protein |
Biological source | Homo sapiens (human) More |
Cellular location | Nucleus: P37231 Nucleus (By similarity): Q15788 |
Total number of polymer chains | 2 |
Total formula weight | 34913.44 |
Authors | Amano, Y. (deposition date: 2011-12-21, release date: 2012-03-07, Last modification date: 2024-03-20) |
Primary citation | Amano, Y.,Yamaguchi, T.,Ohno, K.,Niimi, T.,Orita, M.,Sakashita, H.,Takeuchi, M. Structural basis for telmisartan-mediated partial activation of PPAR gamma Hypertens Res, 35:715-719, 2012 Cited by PubMed: 22357520DOI: 10.1038/hr.2012.17 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.18 Å) |
Structure validation
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