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3RAW

Crystal Structure of human CDC-like kinase 3 isoform in complex with leucettine L41

Summary for 3RAW
Entry DOI10.2210/pdb3raw/pdb
Related2EU9
DescriptorDual specificity protein kinase CLK3, 5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4H-imidazol-4-one (3 entities in total)
Functional Keywordstransferase, kinase, tyrosine-protein kinase, serine/threonine-protein kinase, nucleotide-binding, structural genomics consortium, sgc
Biological sourceHomo sapiens (human)
Cellular locationNucleus: P49761
Total number of polymer chains2
Total formula weight90194.73
Authors
Primary citationFilippakopoulos, P.,Fedorov, O.,King, O.,Bullock, A.,Muniz, J.R.C.,von Delft, F.,Arrowsmith, C.H.,Edwards, A.M.,Weigelt, J.,Bountra, C.,Knapp, S.,Structural Genomics Consortium (SGC)
Crystal Structure of human CDC-like kinase 3 isoform with a benzo-dioxol ligand
To be Published,
Experimental method
X-RAY DIFFRACTION (2.09 Å)
Structure validation

218853

건을2024-04-24부터공개중

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