3QBJ
Crystal structure of dipeptidyl peptidase IV in complex with inhibitor
Summary for 3QBJ
Entry DOI | 10.2210/pdb3qbj/pdb |
Related | 3F8S |
Descriptor | Dipeptidyl peptidase 4, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, alpha-D-mannopyranose-(1-3)-beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... (6 entities in total) |
Functional Keywords | diabetes mellitus, dipeptidyl-peptidase iv inhibitor, hypoglycemic agent, pyrrolidines, sprague-dawley, structure-activity relationship, hydrolase, glycosylation, hydrolase-hydrolase inhibitor complex, hydrolase/hydrolase inhibitor |
Biological source | Homo sapiens (human) |
Total number of polymer chains | 2 |
Total formula weight | 176061.70 |
Authors | Liu, S.P. (deposition date: 2011-01-13, release date: 2012-01-25, Last modification date: 2020-07-29) |
Primary citation | Liu, S.P. Crystal structure of dipeptidyl peptidase IV in complex with inhibitor To be Published, |
Experimental method | X-RAY DIFFRACTION (2.21 Å) |
Structure validation
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