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3OUJ

PHD2 with 2-Oxoglutarate

Summary for 3OUJ
Entry DOI10.2210/pdb3ouj/pdb
Related3OUH 3OUI
DescriptorEgl nine homolog 1, SULFATE ION, FE (II) ION, ... (5 entities in total)
Functional Keywordsphd2, 2og, oxidoreductase
Biological sourceHomo sapiens (human)
Cellular locationCytoplasm : Q9GZT9
Total number of polymer chains1
Total formula weight26877.28
Authors
Staker, B.L.,Arakaki, T.L. (deposition date: 2010-09-14, release date: 2010-12-01, Last modification date: 2024-02-21)
Primary citationRosen, M.D.,Venkatesan, H.,Peltier, H.M.,Bembenek, S.D.,Kanelakis, K.C.,Zhao, L.X.,Leonard, B.E.,Hocutt, F.M.,Wu, X.,Palomino, H.L.,Brondstetter, T.I.,Haugh, P.V.,Cagnon, L.,Yan, W.,Liotta, L.A.,Young, A.,Mirzadegan, T.,Shankley, N.P.,Barrett, T.D.,Rabinowitz, M.H.
Benzimidazole-2-pyrazole HIF Prolyl 4-Hydroxylase Inhibitors as Oral Erythropoietin Secretagogues.
ACS Med Chem Lett, 1:526-529, 2010
Cited by
PubMed: 24900242
DOI: 10.1021/ml100198y
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.3 Å)
Structure validation

217705

數據於2024-03-27公開中

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