Loading
PDBj
メニューPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

3M42

Crystal structure of MAPKAP kinase 2 (MK2) complexed with a tetracyclic ATP site inhibitor

3M42 の概要
エントリーDOI10.2210/pdb3m42/pdb
関連するPDBエントリー3KGA 3M2W
分子名称MAP kinase-activated protein kinase 2, MAGNESIUM ION, 2-[5-(2-methoxyethoxy)pyridin-3-yl]-8,9,10,11-tetrahydro-7H-pyrido[3',4':4,5]pyrrolo[2,3-f]isoquinolin-7-one, ... (4 entities in total)
機能のキーワードsmall molecule inhibitor, atp-site kinase inhibitor, novartis-product nvp-bma086, atp-binding, kinase, nucleotide-binding, phosphoprotein, serine/threonine-protein kinase, transferase
由来する生物種Homo sapiens (human)
タンパク質・核酸の鎖数1
化学式量合計34976.77
構造登録者
Scheufler, C.,Revesz, L.,Be, C.,Izaac, A.,Huppertz, C.,Schlapbach, A.,Kroemer, M. (登録日: 2010-03-10, 公開日: 2011-03-23, 最終更新日: 2024-02-21)
主引用文献Revesz, L.,Schlapbach, A.,Aichholz, R.,Feifel, R.,Hawtin, S.,Heng, R.,Hiestand, P.,Jahnke, W.,Koch, G.,Moebitz, H.,Scheufler, C.,Velcicky, J.,Huppertz, C.
Novel pyrrolo[2,3-f]isoquinoline based MAPKAP-K2 (MK2) inhibitors with potent in vitro and in vivo activity
To be Published,
実験手法
X-RAY DIFFRACTION (2.68 Å)
構造検証レポート
Validation report summary of 3m42
検証レポート(詳細版)ダウンロードをダウンロード

217705

件を2024-03-27に公開中

PDB statisticsPDBj update infoContact PDBjnumon