3KXH
Crystal structure of Z. mays CK2 kinase alpha subunit in complex with the inhibitor (2-dymethylammino-4,5,6,7-tetrabromobenzoimidazol-1yl-acetic acid (K66)
Summary for 3KXH
Entry DOI | 10.2210/pdb3kxh/pdb |
Related | 1zoh 2oxx 3KXG 3KXJ 3KXM 3KXN |
Descriptor | Casein kinase II subunit alpha, [4,5,6,7-tetrabromo-2-(dimethylamino)-1H-benzimidazol-1-yl]acetic acid, DI(HYDROXYETHYL)ETHER, ... (4 entities in total) |
Functional Keywords | protein kinase ck2-inhibitor complex, atp-binding, kinase, nucleotide-binding, serine/threonine-protein kinase, transferase, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
Biological source | Zea mays (maize) |
Total number of polymer chains | 1 |
Total formula weight | 39330.34 |
Authors | Papinutto, E.,Franchin, C.,Battistutta, R. (deposition date: 2009-12-03, release date: 2010-11-17, Last modification date: 2017-11-01) |
Primary citation | Sarno, S.,Papinutto, E.,Franchin, C.,Bain, J.,Elliott, M.,Meggio, F.,Kazimierczuk, Z.,Orzeszko, A.,Zanotti, G.,Battistutta, R.,Pinna, L.A. ATP site-directed inhibitors of protein kinase CK2: an update. Curr Top Med Chem, 11:1340-1351, 2011 Cited by PubMed: 21513497PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.7 Å) |
Structure validation
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