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3KXG

Crystal structure of Z. mays CK2 kinase alpha subunit in complex with the inhibitor 3,4,5,6,7-pentabromo-1H-indazole (K64)

Summary for 3KXG
Entry DOI10.2210/pdb3kxg/pdb
Related1zoh 2oxx 3KXH 3KXJ 3KXM 3KXN
DescriptorCasein kinase II subunit alpha, 3,4,5,6,7-pentabromo-1H-indazole (3 entities in total)
Functional Keywordsprotein kinase ck2-inhibitor complex, atp-binding, kinase, nucleotide-binding, serine/threonine-protein kinase, transferase, transferase-transferase inhibitor complex, transferase/transferase inhibitor
Biological sourceZea mays (maize)
Total number of polymer chains1
Total formula weight39202.01
Authors
Papinutto, E.,Franchin, C.,Battistutta, R. (deposition date: 2009-12-03, release date: 2010-11-17, Last modification date: 2017-11-01)
Primary citationSarno, S.,Papinutto, E.,Franchin, C.,Bain, J.,Elliott, M.,Meggio, F.,Kazimierczuk, Z.,Orzeszko, A.,Zanotti, G.,Battistutta, R.,Pinna, L.A.
ATP site-directed inhibitors of protein kinase CK2: an update.
Curr Top Med Chem, 11:1340-1351, 2011
Cited by
PubMed: 21513497
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.7 Å)
Structure validation

217157

건을2024-03-13부터공개중

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