3KI6
Catalytic fragment of Cholix toxin from Vibrio Cholerae in complex with inhibitor GP-L
Summary for 3KI6
Entry DOI | 10.2210/pdb3ki6/pdb |
Related | 2Q5T 2Q6M 3ESS 3KI0 3KI1 3KI2 3KI3 3KI4 3KI5 3KI7 |
Descriptor | Cholix toxin, 8-fluoro-2-(3-piperidin-1-ylpropanoyl)-1,3,4,5-tetrahydrobenzo[c][1,6]naphthyridin-6(2H)-one (3 entities in total) |
Functional Keywords | adp-ribosyl transferase, alpha-beta complex, diphthamide, transferase, toxin |
Biological source | Vibrio cholerae |
Total number of polymer chains | 1 |
Total formula weight | 23692.26 |
Authors | Jorgensen, R.,Edwards, P.R.,Merrill, A.R. (deposition date: 2009-10-31, release date: 2010-10-27, Last modification date: 2023-09-06) |
Primary citation | Jorgensen, R.,Edwards, P.R.,Merrill, A.R. Structure function analysis of soluble inhibitors of cholix toxin from Vibrio cholerae To be Published, |
Experimental method | X-RAY DIFFRACTION (1.54 Å) |
Structure validation
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