3K6P

Estrogen Related Receptor alpha in Complex with an Ether Based Ligand

3K6P の概要

• エントリーDOI: 10.2210/pdb3k6p/pdb
• 分子名称: Steroid hormone receptor ERR1, 4-(4-{[(5R)-2,4-dioxo-1,3-thiazolidin-5-yl]methyl}-2-methoxyphenoxy)-3-(trifluoromethyl)benzonitrile (3 entities in total)
• 機能のキーワード: estrogen related receptor alpha, dna-binding, isopeptide bond, metal-binding, nucleus, phosphoprotein, receptor, transcription, transcription regulation, zinc-finger, hormone receptor
• 由来する生物種: Homo sapiens (human)
• タンパク質・核酸の鎖数: 1
• 化学式量合計: 27586.74

構造登録者

Abad, M.C.,Patch, R.J. (登録日: 2009-10-09, 公開日: 2010-10-20, 最終更新日: 2023-09-06)

• 主引用文献: Patch, R.J.,Searle, L.L.,Kim, A.J.,De, D.,Zhu, X.,Askari, H.B.,O'Neill, J.C.,Abad, M.C.,Rentzeperis, D.,Geisler, J.G.; Development of Diaryl Ether based ligands for Estrogen Related Receptor alpha as Potential Anti-Diabetic Agents.; To be Published,

実験手法

X-RAY DIFFRACTION (1.996 Å)