3H9R
Crystal structure of the kinase domain of type I activin receptor (ACVR1) in complex with FKBP12 and dorsomorphin
3H9R の概要
エントリーDOI | 10.2210/pdb3h9r/pdb |
分子名称 | Activin receptor type-1, Peptidyl-prolyl cis-trans isomerase FKBP1A, 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine, ... (6 entities in total) |
機能のキーワード | structural genomics, structural genomics consortium, sgc, atp-binding, disease mutation, glycoprotein, kinase, magnesium, manganese, membrane, metal-binding, nucleotide-binding, phosphoprotein, receptor, serine/threonine-protein kinase, transferase, transmembrane, isomerase, rotamase, isomerase-protein kinase complex, isomerase/protein kinase |
由来する生物種 | Homo sapiens (human) 詳細 |
細胞内の位置 | Membrane; Single-pass type I membrane protein: Q04771 Cytoplasm: P62942 |
タンパク質・核酸の鎖数 | 2 |
化学式量合計 | 50916.01 |
構造登録者 | Chaikuad, A.,Alfano, I.,Shrestha, B.,Muniz, J.R.C.,Petrie, K.,Fedorov, O.,Phillips, C.,Bishop, S.,Mahajan, P.,Pike, A.C.W.,von Delft, F.,Arrowsmith, C.H.,Edwards, A.M.,Weigelt, J.,Bountra, C.,Knapp, S.,Bullock, A.,Structural Genomics Consortium (SGC) (登録日: 2009-04-30, 公開日: 2009-06-02, 最終更新日: 2023-09-06) |
主引用文献 | Chaikuad, A.,Alfano, I.,Kerr, G.,Sanvitale, C.E.,Boergermann, J.H.,Triffitt, J.T.,von Delft, F.,Knapp, S.,Knaus, P.,Bullock, A.N. Structure of the Bone Morphogenetic Protein Receptor ALK2 and Implications for Fibrodysplasia Ossificans Progressiva. J.Biol.Chem., 287:36990-36998, 2012 Cited by PubMed: 22977237DOI: 10.1074/jbc.M112.365932 主引用文献が同じPDBエントリー |
実験手法 | X-RAY DIFFRACTION (2.35 Å) |
構造検証レポート
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