3GP0
Crystal Structure of Human Mitogen Activated Protein Kinase 11 (p38 beta) in complex with Nilotinib
3GP0 の概要
エントリーDOI | 10.2210/pdb3gp0/pdb |
分子名称 | Mitogen-activated protein kinase 11, Nilotinib, 1,2-ETHANEDIOL, ... (5 entities in total) |
機能のキーワード | mitogen-activated protein kinase 11, p38b, p38beta, prkm11, sapk2, sapk2b, stress-activated protein kinase-2, structural genomics consortium, sgc, atp-binding, kinase, nucleotide-binding, phosphoprotein, serine/threonine-protein kinase, transferase, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
由来する生物種 | Homo sapiens (human) |
タンパク質・核酸の鎖数 | 1 |
化学式量合計 | 40379.38 |
構造登録者 | Filippakopoulos, P.,Barr, A.,Fedorov, O.,Keates, T.,Soundararajan, M.,Elkins, J.,Salah, E.,Burgess-Brown, N.,Ugochukwu, E.,Pike, A.C.W.,Muniz, J.,Roos, A.,Chaikuad, A.,von Delft, F.,Arrowsmith, C.H.,Edwards, A.M.,Weigelt, J.,Bountra, C.,Knapp, S.,Structural Genomics Consortium (SGC) (登録日: 2009-03-20, 公開日: 2009-04-07, 最終更新日: 2023-09-06) |
主引用文献 | Filippakopoulos, P.,Barr, A.,Fedorov, O.,Keates, T.,Soundararajan, M.,Elkins, J.,Salah, E.,Burgess-Brown, N.,Ugochukwu, E.,Pike, A.C.W.,Muniz, J.,Roos, A.,Chaikuad, A.,von Delft, F.,Arrowsmith, C.H.,Edwards, A.M.,Weigelt, J.,Bountra, C.,Knapp, S.,Structural Genomics Consortium (SGC) Crystal Structure of Human Mitogen Activated Protein Kinase 11 (p38 beta) in complex with Nilotinib To be Published, |
実験手法 | X-RAY DIFFRACTION (1.9 Å) |
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