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3FL5

Protein kinase CK2 in complex with the inhibitor Quinalizarin

Summary for 3FL5
Entry DOI10.2210/pdb3fl5/pdb
Related1F0Q 3BQC
DescriptorCasein kinase II subunit alpha, DI(HYDROXYETHYL)ETHER, 1,2,5,8-tetrahydroxyanthracene-9,10-dione, ... (4 entities in total)
Functional Keywordsprotein kinase ck2-inhibitor complex, atp-binding, kinase, nucleotide-binding, serine/threonine-protein kinase, transferase
Biological sourceZea mays
Total number of polymer chains1
Total formula weight39685.49
Authors
Mazzorana, M.,Franchin, C.,Battistutta, R. (deposition date: 2008-12-18, release date: 2009-08-18, Last modification date: 2017-11-01)
Primary citationCozza, G.,Mazzorana, M.,Papinutto, E.,Bain, J.,Elliott, M.,di Maira, G.,Gianoncelli, A.,Pagano, M.A.,Sarno, S.,Ruzzene, M.,Battistutta, R.,Meggio, F.,Moro, S.,Zagotto, G.,Pinna, L.A.
Quinalizarin as a potent, selective and cell-permeable inhibitor of protein kinase CK2
Biochem.J., 421:387-395, 2009
Cited by
PubMed: 19432557
DOI: 10.1042/BJ20090069
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.3 Å)
Structure validation

217157

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