3BQR
Crystal structure of human death associated protein kinase 3 (DAPK3) in complex with an imidazo-pyridazine ligand
3BQR の概要
エントリーDOI | 10.2210/pdb3bqr/pdb |
分子名称 | Death-associated protein kinase 3, 4-(6-{[(1R)-1-(hydroxymethyl)propyl]amino}imidazo[1,2-b]pyridazin-3-yl)benzoic acid, S-1,2-PROPANEDIOL, ... (5 entities in total) |
機能のキーワード | death associated kinase, dapk3, zip kinase, zipk, dap kinase 3, dap like kinase, dlk, structural genomics consortium, sgc, apoptosis, atp-binding, chromatin regulator, nucleotide-binding, nucleus, serine/threonine-protein kinase, transferase |
由来する生物種 | Homo sapiens (human) |
細胞内の位置 | Nucleus . Isoform 1: Nucleus . Isoform 2: Nucleus : O43293 |
タンパク質・核酸の鎖数 | 1 |
化学式量合計 | 33115.75 |
構造登録者 | Filippakopoulos, P.,Rellos, P.,Fedorov, O.,Niesen, F.,Pike, A.C.W.,Pilka, E.S.,von Delft, F.,Arrowsmith, C.H.,Edwards, A.M.,Weigelt, J.,Knapp, S.,Structural Genomics Consortium (SGC) (登録日: 2007-12-20, 公開日: 2008-02-26, 最終更新日: 2023-08-30) |
主引用文献 | Filippakopoulos, P.,Rellos, P.,Fedorov, O.,Niesen, F.,Pike, A.C.W.,Pilka, E.S.,von Delft, F.,Arrowsmith, C.H.,Edwards, A.M.,Weigelt, J.,Knapp, S. Crystal Structure of Human Death Associated Protein Kinase 3 (DAPK3) in Complex with an Imidazo-Pyridazine Ligand. To be Published, |
実験手法 | X-RAY DIFFRACTION (1.75 Å) |
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