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3BL7

Synthetic Gene Encoded DcpS bound to inhibitor DG156844

Summary for 3BL7
Entry DOI10.2210/pdb3bl7/pdb
Related1ST0 1ST4 3BL9 3BLA
DescriptorScavenger mRNA-decapping enzyme DcpS, 5-{[1-(2-fluorobenzyl)piperidin-4-yl]methoxy}quinazoline-2,4-diamine (3 entities in total)
Functional Keywordsmrna decapping enzyme, dcps, ligand complex, cytoplasm, hydrolase, nonsense-mediated mrna decay, nucleus, polymorphism, structural genomics, psi-2, protein structure initiative, accelerated technologies center for gene to 3d structure, atcg3d
Biological sourceHomo sapiens (Human)
Cellular locationCytoplasm: Q96C86
Total number of polymer chains2
Total formula weight70164.67
Authors
Staker, B.L.,Christensen, J.,Stewart, L.,Accelerated Technologies Center for Gene to 3D Structure (ATCG3D) (deposition date: 2007-12-10, release date: 2008-10-21, Last modification date: 2023-08-30)
Primary citationSingh, J.,Salcius, M.,Liu, S.W.,Staker, B.L.,Mishra, R.,Thurmond, J.,Michaud, G.,Mattoon, D.R.,Printen, J.,Christensen, J.,Bjornsson, J.M.,Pollok, B.A.,Kiledjian, M.,Stewart, L.,Jarecki, J.,Gurney, M.E.
DcpS as a therapeutic target for spinal muscular atrophy.
Acs Chem.Biol., 3:711-722, 2008
Cited by
PubMed: 18839960
DOI: 10.1021/cb800120t
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.31 Å)
Structure validation

217705

數據於2024-03-27公開中

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