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3UYT

crystal structure of ck1d with PF670462 from P1 crystal form

Summary for 3UYT
Entry DOI10.2210/pdb3uyt/pdb
Related1CKI 3UYS 3UZP
DescriptorCasein kinase I isoform delta, 4-[1-cyclohexyl-4-(4-fluorophenyl)-1H-imidazol-5-yl]pyrimidin-2-amine, SULFATE ION, ... (4 entities in total)
Functional Keywordsck1d, kinase, inhibitor, pf670462, transferase-transferase inhibitor complex, transferase/transferase inhibitor
Biological sourceHomo sapiens (human)
Cellular locationCytoplasm: P48730
Total number of polymer chains4
Total formula weight139424.66
Authors
Huang, X. (deposition date: 2011-12-06, release date: 2012-01-11, Last modification date: 2024-02-28)
Primary citationLong, A.,Zhao, H.,Huang, X.
Structural basis for the interaction between casein kinase 1 delta and a potent and selective inhibitor.
J.Med.Chem., 55:956-960, 2012
Cited by
PubMed: 22168824
DOI: 10.1021/jm201387s
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2 Å)
Structure validation

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