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2GPA

ALLOSTERIC INHIBITION OF GLYCOGEN PHOSPHORYLASE A BY A POTENTIAL ANTIDIABETIC DRUG

2GPA の概要
エントリーDOI10.2210/pdb2gpa/pdb
分子名称PROTEIN (GLYCOGEN PHOSPHORYLASE), alpha-D-glucopyranose, PYRIDOXAL-5'-PHOSPHATE, ... (5 entities in total)
機能のキーワードdiabetes, glycogen metabolism, phosphorylase a, inhibition, allosteric site, transferase
由来する生物種Oryctolagus cuniculus (rabbit)
タンパク質・核酸の鎖数1
化学式量合計97890.57
構造登録者
Oikonomakos, N.G.,Tsitsanou, K.E.,Zographos, S.E.,Skamnaki, V.T. (登録日: 1999-02-18, 公開日: 1999-02-26, 最終更新日: 2023-12-27)
主引用文献Oikonomakos, N.G.,Tsitsanou, K.E.,Zographos, S.E.,Skamnaki, V.T.,Goldmann, S.,Bischoff, H.
Allosteric inhibition of glycogen phosphorylase a by the potential antidiabetic drug 3-isopropyl 4-(2-chlorophenyl)-1,4-dihydro-1-ethyl-2-methyl-pyridine-3,5,6-tricarbo xylate.
Protein Sci., 8:1930-1945, 1999
Cited by
PubMed: 10548038
主引用文献が同じPDBエントリー
実験手法
X-RAY DIFFRACTION (2 Å)
構造検証レポート
Validation report summary of 2gpa
検証レポート(詳細版)ダウンロードをダウンロード

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件を2024-03-27に公開中

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