2CSN
BINARY COMPLEX OF CASEIN KINASE-1 WITH CKI7
Summary for 2CSN
Entry DOI | 10.2210/pdb2csn/pdb |
Descriptor | CASEIN KINASE-1, SULFATE ION, N-(2-AMINOETHYL)-5-CHLOROISOQUINOLINE-8-SULFONAMIDE, ... (4 entities in total) |
Functional Keywords | casein kinase-1, protein kinase |
Biological source | Schizosaccharomyces pombe (fission yeast) |
Cellular location | Cytoplasm: P40233 |
Total number of polymer chains | 1 |
Total formula weight | 34723.92 |
Authors | |
Primary citation | Xu, R.M.,Carmel, G.,Kuret, J.,Cheng, X. Structural basis for selectivity of the isoquinoline sulfonamide family of protein kinase inhibitors. Proc.Natl.Acad.Sci.USA, 93:6308-6313, 1996 Cited by PubMed: 8692811DOI: 10.1073/pnas.93.13.6308 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.5 Å) |
Structure validation
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