1STC
CAMP-DEPENDENT PROTEIN KINASE, ALPHA-CATALYTIC SUBUNIT IN COMPLEX WITH STAUROSPORINE
1STC の概要
エントリーDOI | 10.2210/pdb1stc/pdb |
分子名称 | CAMP-DEPENDENT PROTEIN KINASE, PROTEIN KINASE INHIBITOR, STAUROSPORINE, ... (4 entities in total) |
機能のキーワード | protein kinase, staurosporine, camp, phosphorylation, complex (transferase-inhibitor), serine/threonine-protein kinase, complex (transferase-inhibitor) complex, complex (transferase/inhibitor) |
由来する生物種 | Bos taurus (cattle) |
細胞内の位置 | Cytoplasm: P00517 |
タンパク質・核酸の鎖数 | 2 |
化学式量合計 | 43479.34 |
構造登録者 | Prade, L.,Engh, R.A.,Girod, A.,Kinzel, V.,Huber, R.,Bossemeyer, D. (登録日: 1997-10-10, 公開日: 1998-02-25, 最終更新日: 2023-08-09) |
主引用文献 | Prade, L.,Engh, R.A.,Girod, A.,Kinzel, V.,Huber, R.,Bossemeyer, D. Staurosporine-induced conformational changes of cAMP-dependent protein kinase catalytic subunit explain inhibitory potential. Structure, 5:1627-1637, 1997 Cited by PubMed: 9438863DOI: 10.1016/S0969-2126(97)00310-9 主引用文献が同じPDBエントリー |
実験手法 | X-RAY DIFFRACTION (2.3 Å) |
構造検証レポート
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