1Q8U
The Catalytic Subunit of cAMP-dependent Protein Kinase in Complex with Rho-kinase Inhibitor H-1152P
1Q8U の概要
エントリーDOI | 10.2210/pdb1q8u/pdb |
関連するPDBエントリー | 1Q8T 1Q8W |
分子名称 | cAMP-dependent protein kinase, alpha-catalytic subunit, cAMP-dependent protein kinase inhibitor, alpha form, (S)-2-METHYL-1-[(4-METHYL-5-ISOQUINOLINE)SULFONYL]-HOMOPIPERAZINE, ... (5 entities in total) |
機能のキーワード | kinase-inhibitor-complex, phosphotransferase/inhibitor, camp, phosphorylation, serine/threonine-protein kinase, atp-binding, pka, rho-kinase, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
由来する生物種 | Bos taurus (cattle) 詳細 |
細胞内の位置 | Cytoplasm: P00517 |
タンパク質・核酸の鎖数 | 2 |
化学式量合計 | 43973.06 |
構造登録者 | Breitenlechner, C.,Gassel, M.,Hidaka, H.,Kinzel, V.,Huber, R.,Engh, R.A.,Bossemeyer, D. (登録日: 2003-08-22, 公開日: 2003-12-16, 最終更新日: 2011-07-13) |
主引用文献 | Breitenlechner, C.,Gassel, M.,Hidaka, H.,Kinzel, V.,Huber, R.,Engh, R.A.,Bossemeyer, D. Protein kinase A in complex with Rho-kinase inhibitors Y-27632, Fasudil, and H-1152P: structural basis of selectivity. Structure, 11:1595-1607, 2003 Cited by PubMed: 14656443DOI: 10.1016/j.str.2003.11.002 主引用文献が同じPDBエントリー |
実験手法 | X-RAY DIFFRACTION (1.9 Å) |
構造検証レポート
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