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1FKG

DESIGN, SYNTHESIS, AND KINETIC EVALUATION OF HIGH-AFFINITY FKBP LIGANDS, AND THE X-RAY CRYSTAL STRUCTURES OF THEIR COMPLEXES WITH FKBP12

Summary for 1FKG
Entry DOI10.2210/pdb1fkg/pdb
DescriptorFK506 BINDING PROTEIN, 1,3-DIPHENYL-1-PROPYL-1-(3,3-DIMETHYL-1,2-DIOXYPENTYL)-2-PIPERIDINE CARBOXYLATE (3 entities in total)
Functional Keywordscis-trans isomerase
Biological sourceHomo sapiens (human)
Cellular locationCytoplasm, cytosol : P62942
Total number of polymer chains1
Total formula weight12286.09
Authors
Primary citationHolt, D.A.,Luengo, J.I.,Yamashita, D.S.,Oh, H.J.,Konialian, A.L.,Yen, H.K.,Rozamus, L.W.,Brandt, M.,Bossard, M.J.,Levy, M.A.,Eggleston, D.S.,Liang, J.,Schultz, L.W.,Stout, T.J.,Clardy, J.
DESIGN, SYNTHESIS, AND KINETIC EVALUATION OF HIGH-AFFINITY FKBP LIGANDS AND THE X-RAY CRYSTAL-STRUCTURES OF THEIR COMPLEXES WITH FKBP12.
J.Am.Chem.Soc., 115:9925-9938, 1993
Cited by
Experimental method
X-RAY DIFFRACTION (2 Å)
Structure validation

217705

건을2024-03-27부터공개중

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