1CKP
HUMAN CYCLIN DEPENDENT KINASE 2 COMPLEXED WITH THE INHIBITOR PURVALANOL B
Summary for 1CKP
Entry DOI | 10.2210/pdb1ckp/pdb |
Descriptor | PROTEIN (CYCLIN-DEPENDENT PROTEIN KINASE 2), PURVALANOL B, 1,2-ETHANEDIOL, ... (4 entities in total) |
Functional Keywords | protein kinase, cell cycle, phosphorylation, cell division, mitosis, inhibition, hormone-growth factor complex, hormone/growth factor |
Biological source | Homo sapiens (human) |
Total number of polymer chains | 1 |
Total formula weight | 34471.46 |
Authors | Gray, N.S.,Thunnissen, A.M.W.H.,Schultz, P.G.,Kim, S.H. (deposition date: 1998-07-14, release date: 1999-01-13, Last modification date: 2023-08-09) |
Primary citation | Gray, N.S.,Wodicka, L.,Thunnissen, A.M.,Norman, T.C.,Kwon, S.,Espinoza, F.H.,Morgan, D.O.,Barnes, G.,LeClerc, S.,Meijer, L.,Kim, S.H.,Lockhart, D.J.,Schultz, P.G. Exploiting chemical libraries, structure, and genomics in the search for kinase inhibitors. Science, 281:533-538, 1998 Cited by PubMed: 9677190DOI: 10.1126/science.281.5376.533 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.05 Å) |
Structure validation
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