1QUR
HUMAN ALPHA-THROMBIN IN COMPLEX WITH BIVALENT, BENZAMIDINE-BASED SYNTHETIC INHIBITOR
Summary for 1QUR
Entry DOI | 10.2210/pdb1qur/pdb |
Descriptor | HUMAN THROMBIN (ALPHA CHAIN), HUMAN THROMBIN (BETA CHAIN), BIVALENT INHIBITOR (BZA-2 HIRULOG), ... (4 entities in total) |
Functional Keywords | trypsin like serine protease, blood coagulation, hydrolase-hydrolase inhibitor complex, hydrolase/hydrolase inhibitor |
Biological source | Homo sapiens (human) More |
Cellular location | Secreted, extracellular space: P00734 P00734 |
Total number of polymer chains | 3 |
Total formula weight | 35187.25 |
Authors | Renatus, M.,Steinmetzer, T. (deposition date: 1999-07-02, release date: 1999-10-14, Last modification date: 2023-11-15) |
Primary citation | Steinmetzer, T.,Renatus, M.,Kunzel, S.,Eichinger, A.,Bode, W.,Wikstrom, P.,Hauptmann, J.,Sturzebecher, J. Design and evaluation of novel bivalent thrombin inhibitors based on amidinophenylalanines. Eur.J.Biochem., 265:598-605, 1999 Cited by PubMed: 10504391DOI: 10.1046/j.1432-1327.1999.00742.x PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2 Å) |
Structure validation
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