1KCE
E. COLI THYMIDYLATE SYNTHASE MUTANT E58Q IN COMPLEX WITH CB3717 AND 2'-DEOXYURIDINE 5'-MONOPHOSPHATE (DUMP)
Summary for 1KCE
Entry DOI | 10.2210/pdb1kce/pdb |
Descriptor | THYMIDYLATE SYNTHASE, 2'-DEOXYURIDINE 5'-MONOPHOSPHATE, 10-PROPARGYL-5,8-DIDEAZAFOLIC ACID, ... (4 entities in total) |
Functional Keywords | transferase, reaction intermediate |
Biological source | Escherichia coli |
Cellular location | Cytoplasm: P0A884 |
Total number of polymer chains | 2 |
Total formula weight | 62690.63 |
Authors | Sage, C.R.,Rutenber, E.E.,Stout, T.J.,Stroud, R.M. (deposition date: 1996-10-22, release date: 1997-04-21, Last modification date: 2024-06-05) |
Primary citation | Sage, C.R.,Rutenber, E.E.,Stout, T.J.,Stroud, R.M. An essential role for water in an enzyme reaction mechanism: the crystal structure of the thymidylate synthase mutant E58Q. Biochemistry, 35:16270-16281, 1996 Cited by PubMed: 8973201DOI: 10.1021/bi961269r PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2 Å) |
Structure validation
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