Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

1IS0

Crystal Structure of a Complex of the Src SH2 Domain with Conformationally Constrained Peptide Inhibitor

Summary for 1IS0
Entry DOI10.2210/pdb1is0/pdb
Related PRD IDPRD_000345
DescriptorTyrosine-protein kinase transforming protein SRC, AY0 GLU GLU ILE peptide (3 entities in total)
Functional Keywordsconformationaly constrained inhibitor, transferase-transferase inhibitor complex, transferase/transferase inhibitor
Biological sourceRous sarcoma virus
More
Total number of polymer chains4
Total formula weight25746.68
Authors
Davidson, J.P.,Lubman, O.,Rose, T.,Waksman, G.,Martin, S.F. (deposition date: 2001-11-02, release date: 2002-02-06, Last modification date: 2023-12-27)
Primary citationDavidson, J.P.,Lubman, O.,Rose, T.,Waksman, G.,Martin, S.F.
Calorimetric and structural studies of 1,2,3-trisubstituted cyclopropanes as conformationally constrained peptide inhibitors of Src SH2 domain binding.
J.Am.Chem.Soc., 124:205-215, 2002
Cited by
PubMed: 11782172
DOI: 10.1021/ja011746f
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.9 Å)
Structure validation

217705

PDB entries from 2024-03-27

PDB statisticsPDBj update infoContact PDBjnumon