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1E8Z

Structure determinants of phosphoinositide 3-kinase inhibition by wortmannin, LY294002, quercetin, myricetin and staurosporine

Summary for 1E8Z
Entry DOI10.2210/pdb1e8z/pdb
Related1E8Y
DescriptorPHOSPHATIDYLINOSITOL 3-KINASE CATALYTIC SUBUNIT, STAUROSPORINE (3 entities in total)
Functional Keywordstransferase, phosphoinositide 3-kinase gamma, secondary messenger generation, pi3k, pi 3k, staurosporine
Biological sourceHOMO SAPIENS (HUMAN)
Total number of polymer chains1
Total formula weight111222.70
Authors
Walker, E.H.,Pacold, M.E.,Perisic, O.,Stephens, L.,Hawkins, P.T.,Wymann, M.P.,Williams, R.L. (deposition date: 2000-10-03, release date: 2000-11-17, Last modification date: 2023-12-13)
Primary citationWalker, E.H.,Pacold, M.E.,Perisic, O.,Stephens, L.,Hawkins, P.T.,Whymann, M.P.,Williams, R.L.
Structural Determinations of Phosphoinositide 3-Kinase Inhibition by Wortmannin, Ly294002, Quercetin, Myricetin and Staurosporine
Mol.Cell, 6:909-, 2000
Cited by
PubMed: 11090628
DOI: 10.1016/S1097-2765(05)00089-4
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.4 Å)
Structure validation

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