2WIH
STRUCTURE OF CDK2-CYCLIN A WITH PHA-848125
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | A, C | CELL DIVISION PROTEIN KINASE 2 | polymer | 309 | 35251.9 | 2 | UniProt (P24941) Pfam (PF00069) In PDB | HOMO SAPIENS (HUMAN) | P33 PROTEIN KINASE |
2 | B, D | CYCLIN-A2 | polymer | 265 | 30279.0 | 2 | UniProt (P20248) Pfam (PF00134) Pfam (PF02984) In PDB | HOMO SAPIENS (HUMAN) | CYCLIN A, CYCLIN A2 |
3 | A, C | N,1,4,4-TETRAMETHYL-8-{[4-(4-METHYLPIPERAZIN-1-YL)PHENYL]AMINO}-4,5-DIHYDRO-1H-PYRAZOLO[4,3-H]QUINAZOLINE-3-CARBOXAMIDE | non-polymer | 460.6 | 2 | Chemie (P48) | |||
4 | D | SULFATE ION | non-polymer | 96.1 | 1 | Chemie (SO4) | |||
5 | water | water | 18.0 | 214 | Chemie (HOH) |
Sequence modifications
A, C: 1 - 298 (UniProt: P24941)
B, D: 173 - 432 (UniProt: P20248)
PDB | External Database | Details |
---|---|---|
Gly -4 | - | expression tag |
Pro -3 | - | expression tag |
Leu -2 | - | expression tag |
Val -1 | - | expression tag |
Asp 0 | - | expression tag |
Glu 299 | - | expression tag |
Arg 300 | - | expression tag |
Pro 301 | - | expression tag |
His 302 | - | expression tag |
Arg 303 | - | expression tag |
Asp 304 | - | expression tag |
PDB | External Database | Details |
---|---|---|
Gly 168 | - | expression tag |
Pro 169 | - | expression tag |
Leu 170 | - | expression tag |
Gly 171 | - | expression tag |
Ser 172 | - | expression tag |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 4 |
Total formula weight | 131061.7 | |
Non-Polymers* | Number of molecules | 3 |
Total formula weight | 1017.2 | |
All* | Total formula weight | 132078.9 |