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5RJJ
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BU of 5rjj by Molmil
PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with NCL-00023833
Descriptor: 4-bromanyl-1,8-naphthyridine, PH-interacting protein
Authors:Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C.
Deposit date:2020-06-02
Release date:2020-06-17
Method:X-RAY DIFFRACTION (1.151 Å)
Cite:PanDDA analysis group deposition of ground-state model
To Be Published
5RJT
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BU of 5rjt by Molmil
PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z404993336
Descriptor: 5-methyl-N-(1-methyl-1H-pyrazol-4-yl)-1,2-oxazole-3-carboxamide, PH-interacting protein
Authors:Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C.
Deposit date:2020-06-02
Release date:2020-06-17
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (1.169 Å)
Cite:PanDDA analysis group deposition of ground-state model
To Be Published
5RJK
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BU of 5rjk by Molmil
PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with NCL-00024661
Descriptor: 5-bromo-2-hydroxybenzonitrile, PH-interacting protein
Authors:Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C.
Deposit date:2020-06-02
Release date:2020-06-17
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (1.21 Å)
Cite:PanDDA analysis group deposition of ground-state model
To Be Published
5RJO
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BU of 5rjo by Molmil
PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with NCL-00023827
Descriptor: 6-bromo-1,3-dihydro-2H-indol-2-one, PH-interacting protein
Authors:Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C.
Deposit date:2020-06-02
Release date:2020-06-17
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (1.22 Å)
Cite:PanDDA analysis group deposition of ground-state model
To Be Published
5RKN
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BU of 5rkn by Molmil
PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z373768900
Descriptor: N-(1-ethyl-1H-pyrazol-4-yl)cyclobutanecarboxamide, PH-interacting protein
Authors:Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C.
Deposit date:2020-06-02
Release date:2020-06-17
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (1.23 Å)
Cite:PanDDA analysis group deposition of ground-state model
To Be Published
5RK2
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BU of 5rk2 by Molmil
PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z54633859
Descriptor: 2-[methyl(pyridin-2-yl)amino]ethan-1-ol, PH-interacting protein
Authors:Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C.
Deposit date:2020-06-02
Release date:2020-06-17
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (1.235 Å)
Cite:PanDDA analysis group deposition of ground-state model
To Be Published
5RKD
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BU of 5rkd by Molmil
PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z2168282707
Descriptor: (6S)-1-methyl-4,5,6,7-tetrahydro-1H-benzotriazole-6-carboxylic acid, PH-interacting protein
Authors:Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C.
Deposit date:2020-06-02
Release date:2020-06-17
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (1.237 Å)
Cite:PanDDA analysis group deposition of ground-state model
To Be Published
5RKS
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BU of 5rks by Molmil
PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z1696844792
Descriptor: 1-(diphenylmethyl)azetidin-3-ol, PH-interacting protein
Authors:Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C.
Deposit date:2020-06-02
Release date:2020-06-17
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (1.24 Å)
Cite:PanDDA analysis group deposition of ground-state model
To Be Published
5RK0
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BU of 5rk0 by Molmil
PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z30932204
Descriptor: N-[(4-sulfamoylphenyl)methyl]acetamide, PH-interacting protein
Authors:Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C.
Deposit date:2020-06-02
Release date:2020-06-17
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (1.24 Å)
Cite:PanDDA analysis group deposition of ground-state model
To Be Published
5RKX
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BU of 5rkx by Molmil
PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z1324080698
Descriptor: 3-fluoro-5-methylbenzene-1-sulfonamide, PH-interacting protein
Authors:Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C.
Deposit date:2020-06-02
Release date:2020-06-17
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (1.24 Å)
Cite:PanDDA analysis group deposition of ground-state model
To Be Published
5RKC
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BU of 5rkc by Molmil
PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z234898257
Descriptor: N-methyl-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)methanamine, PH-interacting protein
Authors:Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C.
Deposit date:2020-06-02
Release date:2020-06-17
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (1.24 Å)
Cite:PanDDA analysis group deposition of ground-state model
To Be Published
5RK6
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BU of 5rk6 by Molmil
PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z198194394
Descriptor: 4-(4-fluorophenyl)piperazine-1-carboxamide, PH-interacting protein
Authors:Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C.
Deposit date:2020-06-02
Release date:2020-06-17
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (1.241 Å)
Cite:PanDDA analysis group deposition of ground-state model
To Be Published
5RKT
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BU of 5rkt by Molmil
PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z1266933824
Descriptor: (1H-pyrazol-4-yl)(pyrrolidin-1-yl)methanone, PH-interacting protein
Authors:Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C.
Deposit date:2020-06-02
Release date:2020-06-17
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (1.241 Å)
Cite:PanDDA analysis group deposition of ground-state model
To Be Published
5RJP
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BU of 5rjp by Molmil
PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with NCL-00024672
Descriptor: 4-bromo-1-(2-hydroxyethyl)pyridin-2(1H)-one, PH-interacting protein
Authors:Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C.
Deposit date:2020-06-02
Release date:2020-06-17
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (1.242 Å)
Cite:PanDDA analysis group deposition of ground-state model
To Be Published
5RKW
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BU of 5rkw by Molmil
PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z27678561
Descriptor: N-(6-methoxy-1,3-benzothiazol-2-yl)cyclopropanecarboxamide, PH-interacting protein
Authors:Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C.
Deposit date:2020-06-02
Release date:2020-06-17
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (1.242 Å)
Cite:PanDDA analysis group deposition of ground-state model
To Be Published
5RK5
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BU of 5rk5 by Molmil
PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z57478994
Descriptor: 5-(methoxymethyl)-1,3,4-thiadiazol-2-amine, PH-interacting protein
Authors:Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C.
Deposit date:2020-06-02
Release date:2020-06-17
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (1.243 Å)
Cite:PanDDA analysis group deposition of ground-state model
To Be Published
5RJY
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BU of 5rjy by Molmil
PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z383325512
Descriptor: N-[(1H-pyrazol-4-yl)methyl]acetamide, PH-interacting protein
Authors:Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C.
Deposit date:2020-06-02
Release date:2020-06-17
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (1.25 Å)
Cite:PanDDA analysis group deposition of ground-state model
To Be Published
5RKH
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BU of 5rkh by Molmil
PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z31432917
Descriptor: 2-(4-methylphenoxy)-1-(4-methylpiperazin-4-ium-1-yl)ethanone, PH-interacting protein
Authors:Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C.
Deposit date:2020-06-02
Release date:2020-06-17
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (1.252 Å)
Cite:PanDDA analysis group deposition of ground-state model
To Be Published
5RKF
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BU of 5rkf by Molmil
PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z1674937530
Descriptor: 2-(1-ethyl-1H-pyrazol-4-yl)ethan-1-ol, PH-interacting protein
Authors:Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C.
Deposit date:2020-06-02
Release date:2020-06-17
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (1.264 Å)
Cite:PanDDA analysis group deposition of ground-state model
To Be Published
5RKI
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BU of 5rki by Molmil
PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z198194396
Descriptor: 4-(furan-2-carbonyl)piperazine-1-carboxamide, PH-interacting protein
Authors:Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C.
Deposit date:2020-06-02
Release date:2020-06-17
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (1.268 Å)
Cite:PanDDA analysis group deposition of ground-state model
To Be Published
5RJR
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BU of 5rjr by Molmil
PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z45705015
Descriptor: PH-interacting protein, ~{N}-[2-(4-fluorophenyl)ethyl]methanesulfonamide
Authors:Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C.
Deposit date:2020-06-02
Release date:2020-06-17
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (1.27 Å)
Cite:PanDDA analysis group deposition of ground-state model
To Be Published
5RK1
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BU of 5rk1 by Molmil
PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z1507502062
Descriptor: 6-methoxy-1,3,4,5-tetrahydro-2H-1-benzazepin-2-one, PH-interacting protein
Authors:Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C.
Deposit date:2020-06-02
Release date:2020-06-17
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (1.271 Å)
Cite:PanDDA analysis group deposition of ground-state model
To Be Published
5RK8
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BU of 5rk8 by Molmil
PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z53116498
Descriptor: 3-(2-methyl-1H-benzimidazol-1-yl)propanamide, PH-interacting protein
Authors:Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C.
Deposit date:2020-06-02
Release date:2020-06-17
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (1.272 Å)
Cite:PanDDA analysis group deposition of ground-state model
To Be Published
5RJZ
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BU of 5rjz by Molmil
PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z755044716
Descriptor: N-ethyl-1H-1,2,3-triazole-4-carboxamide, PH-interacting protein
Authors:Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C.
Deposit date:2020-06-02
Release date:2020-06-17
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (1.275 Å)
Cite:PanDDA analysis group deposition of ground-state model
To Be Published
5RKV
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BU of 5rkv by Molmil
PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z56877838
Descriptor: 2-(4-ethoxyphenyl)ethanoic acid, PH-interacting protein
Authors:Grosjean, H, Aimon, A, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Arrowsmith, C.H, Edwards, A, Bountra, C, von Delft, F, Biggin, P.C.
Deposit date:2020-06-02
Release date:2020-06-17
Last modified:2024-03-06
Method:X-RAY DIFFRACTION (1.277 Å)
Cite:PanDDA analysis group deposition of ground-state model
To Be Published

 

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