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6O0L

crystal structure of BCL-2 G101V mutation with venetoclax

GO(遺伝子オントロジー)由来の情報
鎖名GO(遺伝子オントロジー)id名前空間内容
A0042981biological_processregulation of apoptotic process
A0043066biological_processnegative regulation of apoptotic process
C0042981biological_processregulation of apoptotic process
C0043066biological_processnegative regulation of apoptotic process
PDBデータベースに由来する情報
site_idAC1
残基数17
詳細binding site for residue LBM A 301
鎖名残基
AARG12
AALA149
AGLU152
APHE153
AVAL156
APHE198
ATYR202
APEG303
AHOH403
AALA100
AASP103
AARG107
ATYR108
ALEU137
ATRP144
AGLY145
AVAL148

site_idAC2
残基数3
詳細binding site for residue PEG A 302
鎖名残基
AARG12
AMET16
APEG303

site_idAC3
残基数5
詳細binding site for residue PEG A 303
鎖名残基
AASN143
ATHR178
ALBM301
APEG302
ACL304

site_idAC4
残基数4
詳細binding site for residue CL A 304
鎖名残基
AGLU179
AASN182
AARG183
APEG303

site_idAC5
残基数19
詳細binding site for residue LBM C 301
鎖名残基
CARG12
CALA100
CASP103
CARG107
CTYR108
CGLU136
CLEU137
CTRP144
CGLY145
CVAL148
CALA149
CGLU152
CPHE153
CVAL156
CPHE198
CTYR202
CPEG303
CHOH401
CHOH404

site_idAC6
残基数2
詳細binding site for residue PEG C 302
鎖名残基
CARG12
CPEG303

site_idAC7
残基数6
詳細binding site for residue PEG C 303
鎖名残基
CARG12
CASN143
CARG146
CLBM301
CPEG302
CCL304

site_idAC8
残基数4
詳細binding site for residue CL C 304
鎖名残基
CGLU179
CASN182
CARG183
CPEG303

UniProtにおけるモチーフ・データベースPROSITEからの機能情報
site_idPS01080
残基数19
詳細BH1 Apoptosis regulator, Bcl-2 family BH1 motif signature. LFrDGv.NWGRIVAFFeFGG
鎖名残基詳細
ALEU137-GLY155

site_idPS01258
残基数12
詳細BH2 Apoptosis regulator, Bcl-2 family BH2 motif signature. WIqdnGGWDaFV
鎖名残基詳細
ATRP188-VAL199

site_idPS01260
残基数21
詳細BH4_1 Apoptosis regulator, Bcl-2 family BH4 motif signature. DNREIVmKYIHYKLSQRGYeW
鎖名残基詳細
AASP10-TRP30

SwissProt/UniProtに記載されている蛋白質分子機能情報
site_idSWS_FT_FI1
残基数2
詳細SITE: Cleavage; by caspase-3
鎖名残基詳細
AASP75
CASP75

225158

件を2024-09-18に公開中

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