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4O0A

Fragment-Based Discovery of a Potent Inhibitor of Replication Protein A Protein-Protein Interactions

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0005634cellular_componentnucleus
A0006260biological_processDNA replication
Functional Information from PDB Data
site_idAC1
Number of Residues21
DetailsBINDING SITE FOR RESIDUE 2P9 A 201
ChainResidue
AARG31
ATHR60
AASN85
AARG91
AVAL93
AILE95
AMET97
AHOH315
AHOH317
AHOH356
AHOH376
AILE33
AHOH415
AHOH438
ATHR34
AARG41
AARG43
ASER54
ASER55
AMET57
AALA59

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsMOD_RES: N-acetylmethionine => ECO:0007744|PubMed:19413330, ECO:0007744|PubMed:22223895
ChainResidueDetails
AMET1

site_idSWS_FT_FI2
Number of Residues3
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin) => ECO:0000269|PubMed:26474068
ChainResidueDetails
ALYS22
ALYS88

218853

數據於2024-04-24公開中

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