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2FNT

Crystal structure of a drug-resistant (V82A) inactive (D25N) HIV-1 protease complexed with AP2V variant of HIV-1 NC-p1 substrate.

GO(遺伝子オントロジー)由来の情報
鎖名GO(遺伝子オントロジー)id名前空間内容
A0004190molecular_functionaspartic-type endopeptidase activity
A0006508biological_processproteolysis
B0004190molecular_functionaspartic-type endopeptidase activity
B0006508biological_processproteolysis
PDBデータベースに由来する情報
site_idAC1
残基数7
詳細BINDING SITE FOR RESIDUE PO4 B 501
鎖名残基
APRO1
BGLY68
BHIS69
BLYS70
BHOH519
BHOH537
BHOH572

site_idAC2
残基数4
詳細BINDING SITE FOR RESIDUE PO4 B 502
鎖名残基
BASN83
BHOH554
BLYS20
BGLU21

site_idAC3
残基数3
詳細BINDING SITE FOR RESIDUE ACT A 504
鎖名残基
ALYS7
AARG8
BARG87

site_idAC4
残基数4
詳細BINDING SITE FOR RESIDUE PO4 A 505
鎖名残基
ALYS20
AGLU21
AASN83
AHOH539

site_idAC5
残基数7
詳細BINDING SITE FOR RESIDUE PO4 A 506
鎖名残基
ATRP6
AGLY51
AHOH571
BTHR91
BGLY94
BHOH512
BHOH521

site_idAC6
残基数8
詳細BINDING SITE FOR RESIDUE PO4 A 507
鎖名残基
AGLY16
APRO63
AHOH546
BGLY16
BGLY17
BHOH520
BHOH530
BHOH585

site_idAC7
残基数5
詳細BINDING SITE FOR RESIDUE PO4 B 508
鎖名残基
BLEU19
BPRO44
BLYS45
BMET46
BHOH586

site_idAC8
残基数2
詳細BINDING SITE FOR RESIDUE ACT B 509
鎖名残基
BLYS7
BARG8

site_idAC9
残基数3
詳細BINDING SITE FOR RESIDUE ACT A 510
鎖名残基
AGLN58
AHOH563
BGLN61

SwissProt/UniProtに記載されている蛋白質分子機能情報
site_idSWS_FT_FI1
残基数2
詳細ACT_SITE: For protease activity; shared with dimeric partner => ECO:0000255|PROSITE-ProRule:PRU10094
鎖名残基詳細
AASN25
BASN25

site_idSWS_FT_FI2
残基数2
詳細SITE: Cleavage; by viral protease => ECO:0000250
鎖名残基詳細
APHE99
BPHE99

218853

件を2024-04-24に公開中

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