2FNT
Crystal structure of a drug-resistant (V82A) inactive (D25N) HIV-1 protease complexed with AP2V variant of HIV-1 NC-p1 substrate.
GO(遺伝子オントロジー)由来の情報
鎖名 | GO(遺伝子オントロジー)id | 名前空間 | 内容 |
A | 0004190 | molecular_function | aspartic-type endopeptidase activity |
A | 0006508 | biological_process | proteolysis |
B | 0004190 | molecular_function | aspartic-type endopeptidase activity |
B | 0006508 | biological_process | proteolysis |
PDBデータベースに由来する情報
site_id | AC1 |
残基数 | 7 |
詳細 | BINDING SITE FOR RESIDUE PO4 B 501 |
鎖名 | 残基 |
A | PRO1 |
B | GLY68 |
B | HIS69 |
B | LYS70 |
B | HOH519 |
B | HOH537 |
B | HOH572 |
site_id | AC2 |
残基数 | 4 |
詳細 | BINDING SITE FOR RESIDUE PO4 B 502 |
鎖名 | 残基 |
B | ASN83 |
B | HOH554 |
B | LYS20 |
B | GLU21 |
site_id | AC3 |
残基数 | 3 |
詳細 | BINDING SITE FOR RESIDUE ACT A 504 |
site_id | AC4 |
残基数 | 4 |
詳細 | BINDING SITE FOR RESIDUE PO4 A 505 |
鎖名 | 残基 |
A | LYS20 |
A | GLU21 |
A | ASN83 |
A | HOH539 |
site_id | AC5 |
残基数 | 7 |
詳細 | BINDING SITE FOR RESIDUE PO4 A 506 |
鎖名 | 残基 |
A | TRP6 |
A | GLY51 |
A | HOH571 |
B | THR91 |
B | GLY94 |
B | HOH512 |
B | HOH521 |
site_id | AC6 |
残基数 | 8 |
詳細 | BINDING SITE FOR RESIDUE PO4 A 507 |
鎖名 | 残基 |
A | GLY16 |
A | PRO63 |
A | HOH546 |
B | GLY16 |
B | GLY17 |
B | HOH520 |
B | HOH530 |
B | HOH585 |
site_id | AC7 |
残基数 | 5 |
詳細 | BINDING SITE FOR RESIDUE PO4 B 508 |
鎖名 | 残基 |
B | LEU19 |
B | PRO44 |
B | LYS45 |
B | MET46 |
B | HOH586 |
site_id | AC8 |
残基数 | 2 |
詳細 | BINDING SITE FOR RESIDUE ACT B 509 |
site_id | AC9 |
残基数 | 3 |
詳細 | BINDING SITE FOR RESIDUE ACT A 510 |
SwissProt/UniProtに記載されている蛋白質分子機能情報
site_id | SWS_FT_FI2 |
残基数 | 2 |
詳細 | SITE: Cleavage; by viral protease => ECO:0000250 |