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1W85

The crystal structure of pyruvate dehydrogenase E1 bound to the peripheral subunit binding domain of E2

GO(遺伝子オントロジー)由来の情報
鎖名GO(遺伝子オントロジー)id名前空間内容
A0004739molecular_functionpyruvate dehydrogenase (acetyl-transferring) activity
A0005515molecular_functionprotein binding
A0009083biological_processbranched-chain amino acid catabolic process
A0016491molecular_functionoxidoreductase activity
A0016624molecular_functionoxidoreductase activity, acting on the aldehyde or oxo group of donors, disulfide as acceptor
B0003824molecular_functioncatalytic activity
B0004739molecular_functionpyruvate dehydrogenase (acetyl-transferring) activity
B0005515molecular_functionprotein binding
B0016491molecular_functionoxidoreductase activity
C0004739molecular_functionpyruvate dehydrogenase (acetyl-transferring) activity
C0005515molecular_functionprotein binding
C0009083biological_processbranched-chain amino acid catabolic process
C0016491molecular_functionoxidoreductase activity
C0016624molecular_functionoxidoreductase activity, acting on the aldehyde or oxo group of donors, disulfide as acceptor
D0003824molecular_functioncatalytic activity
D0004739molecular_functionpyruvate dehydrogenase (acetyl-transferring) activity
D0005515molecular_functionprotein binding
D0016491molecular_functionoxidoreductase activity
E0004739molecular_functionpyruvate dehydrogenase (acetyl-transferring) activity
E0005515molecular_functionprotein binding
E0009083biological_processbranched-chain amino acid catabolic process
E0016491molecular_functionoxidoreductase activity
E0016624molecular_functionoxidoreductase activity, acting on the aldehyde or oxo group of donors, disulfide as acceptor
F0003824molecular_functioncatalytic activity
F0004739molecular_functionpyruvate dehydrogenase (acetyl-transferring) activity
F0005515molecular_functionprotein binding
F0016491molecular_functionoxidoreductase activity
G0004739molecular_functionpyruvate dehydrogenase (acetyl-transferring) activity
G0005515molecular_functionprotein binding
G0009083biological_processbranched-chain amino acid catabolic process
G0016491molecular_functionoxidoreductase activity
G0016624molecular_functionoxidoreductase activity, acting on the aldehyde or oxo group of donors, disulfide as acceptor
H0003824molecular_functioncatalytic activity
H0004739molecular_functionpyruvate dehydrogenase (acetyl-transferring) activity
H0005515molecular_functionprotein binding
H0016491molecular_functionoxidoreductase activity
I0016746molecular_functionacyltransferase activity
J0016746molecular_functionacyltransferase activity
PDBデータベースに由来する情報
site_idAC1
残基数4
詳細BINDING SITE FOR RESIDUE MG A1368
鎖名残基
AASP173
AASN202
APHE204
ATPP1370

site_idAC2
残基数6
詳細BINDING SITE FOR RESIDUE K B1325
鎖名残基
BHOH2069
BILE112
BTHR113
BALA160
BASP163
BASP165

site_idAC3
残基数6
詳細BINDING SITE FOR RESIDUE MG B1326
鎖名残基
AHOH2131
BHOH2045
BHOH2046
CHOH2169
CHOH2170
DHOH2071

site_idAC4
残基数5
詳細BINDING SITE FOR RESIDUE MG C1368
鎖名残基
CASP173
CASN202
CPHE204
CTPP1370
CHOH2173

site_idAC5
残基数6
詳細BINDING SITE FOR RESIDUE K D1325
鎖名残基
DILE112
DTHR113
DALA160
DASP163
DASP165
DHOH2087

site_idAC6
残基数5
詳細BINDING SITE FOR RESIDUE MG E1368
鎖名残基
EASP173
EASN202
ETPP1370
EHOH2079
EHOH2087

site_idAC7
残基数6
詳細BINDING SITE FOR RESIDUE K F1325
鎖名残基
FILE112
FTHR113
FALA160
FASP163
FASP165
FHOH2060

site_idAC8
残基数6
詳細BINDING SITE FOR RESIDUE MG F1326
鎖名残基
EHOH2083
EHOH2084
FHOH2045
GHOH2125
GHOH2127
HHOH2057

site_idAC9
残基数5
詳細BINDING SITE FOR RESIDUE MG G1368
鎖名残基
GASP173
GASN202
GPHE204
GTPP1370
GHOH2131

site_idBC1
残基数6
詳細BINDING SITE FOR RESIDUE K H1325
鎖名残基
HILE112
HTHR113
HALA160
HASP163
HASP165
HHOH2072

site_idBC2
残基数25
詳細BINDING SITE FOR RESIDUE TDP A1370
鎖名残基
ATYR102
AARG103
AILE142
AILE143
AILE144
AGLY172
AASP173
AGLY174
AGLY175
AGLN178
AASN202
APHE204
AALA205
AILE206
AHIS271
AMG1368
AHOH2163
AHOH2222
AHOH2223
AHOH2224
DGLU28
DLEU57
DGLU59
DGLN81
DPHE85

site_idBC3
残基数26
詳細BINDING SITE FOR RESIDUE TDP C1370
鎖名残基
CHIS271
CMG1368
CHOH2173
CHOH2279
CHOH2280
CHOH2281
CHOH2282
BGLU28
BLEU57
BGLU59
BGLN81
BPHE85
CTYR102
CARG103
CILE142
CILE143
CILE144
CGLY172
CASP173
CGLY174
CGLY175
CGLN178
CASN202
CPHE204
CALA205
CILE206

site_idBC4
残基数20
詳細BINDING SITE FOR RESIDUE TDP E1370
鎖名残基
ETYR102
EARG103
EILE142
EILE144
EGLY172
EASP173
EGLY174
EGLY175
EGLN178
EASN202
EHIS271
EMG1368
EHOH2087
EHOH2136
EHOH2137
HGLU28
HLEU57
HGLU59
HGLN81
HPHE85

site_idBC5
残基数25
詳細BINDING SITE FOR RESIDUE TDP G1370
鎖名残基
FGLU28
FLEU57
FGLU59
FGLN81
FPHE85
GTYR102
GARG103
GILE142
GILE144
GGLY172
GASP173
GGLY174
GGLY175
GGLN178
GASN202
GPHE204
GALA205
GILE206
GHIS271
GMG1368
GHOH2131
GHOH2231
GHOH2232
GHOH2233
GHOH2234

site_idBC6
残基数3
詳細BINDING SITE FOR RESIDUE PEG A1369
鎖名残基
AMET160
APHE191
BGLU49

site_idBC7
残基数4
詳細BINDING SITE FOR RESIDUE PEG C1369
鎖名残基
CMET160
CPHE191
CHOH2152
DGLU49

site_idBC8
残基数3
詳細BINDING SITE FOR RESIDUE PEG G1369
鎖名残基
GILE109
GTRP110
GGLU324

SwissProt/UniProtに記載されている蛋白質分子機能情報
site_idSWS_FT_FI1
残基数4
詳細BINDING: BINDING => ECO:0000250
鎖名残基詳細
BSER60
DSER60
FSER60
HSER60

CSAにおける酵素触媒機能の情報
site_idCSA1
残基数3
詳細Annotated By Reference To The Literature 1dtw
鎖名残基詳細
CHIS271
BGLU59
BHIS128

site_idCSA2
残基数3
詳細Annotated By Reference To The Literature 1dtw
鎖名残基詳細
AHIS271
DGLU59
DHIS128

site_idCSA3
残基数3
詳細Annotated By Reference To The Literature 1dtw
鎖名残基詳細
FGLU59
FHIS128
GHIS271

site_idCSA4
残基数3
詳細Annotated By Reference To The Literature 1dtw
鎖名残基詳細
HGLU59
HHIS128
EHIS271

site_idMCSA1
残基数2
詳細M-CSA 106
鎖名残基詳細
BSER60proton acceptor, proton donor
BSER129proton acceptor, proton donor
AARG282electrostatic stabiliser, hydrogen bond donor

site_idMCSA2
残基数2
詳細M-CSA 106
鎖名残基詳細
DSER60proton acceptor, proton donor
DSER129proton acceptor, proton donor
CARG282electrostatic stabiliser, hydrogen bond donor

site_idMCSA3
残基数2
詳細M-CSA 106
鎖名残基詳細
FSER60proton acceptor, proton donor
FSER129proton acceptor, proton donor
EARG282electrostatic stabiliser, hydrogen bond donor

site_idMCSA4
残基数2
詳細M-CSA 106
鎖名残基詳細
HSER60proton acceptor, proton donor
HSER129proton acceptor, proton donor
GARG282electrostatic stabiliser, hydrogen bond donor

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件を2024-09-18に公開中

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