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1DIF

HIV-1 PROTEASE IN COMPLEX WITH A DIFLUOROKETONE CONTAINING INHIBITOR A79285

Experimental procedure
Detector technologyIMAGE PLATE
DetectorRIGAKU
Spacegroup nameP 21 21 21
格子定数 [Å]52.000, 59.900, 62.100
格子定数 [度]90.00, 90.00, 90.00
精密化法
残基10.000 - 1.700
R因子0.198
Rwork0.198
結合長の平均二乗偏差(RMSD) [Å]0.017
結合角の平均二乗偏差(RMSD) [度]29.100

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Data reduction softwareMOSFLM
Phasing softwareX-PLOR
Refinement softwareX-PLOR
Quality characteristics
 Overall
分解能 [Å] (高)1.700

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Rmerge_l_obs0.092

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Total number of observations40709

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独立反射数20479
完全性 [%]94.9
冗長性2
結晶化条件
結晶ID方法pH温度溶液条件
1Vapor diffusion, hanging drop

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6.2

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文献の結晶化試薬
ID結晶ID溶液試薬名濃度 (単位) (単位)詳細
11dropprotease8 (mg/ml)
21dropsodium acetate50 (mM)
31dropdithiothreitol10 (mM)
41reservoirammonium sulfate37 (%(w/v))
51reservoircitrate63 (mM)
61reservoirsodium phosphate126 (mM)
71reservoirbeta-mercaptoethanol1 (M)
81reservoirdimethyl sulfoxide
91reservoirisopropanol

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件を2024-09-18に公開中

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