- PDB-4ly9: Human GKRP complexed to AMG-1694 [(2R)-1,1,1-trifluoro-2-{4-[(2S)... -
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基本情報
登録情報
データベース: PDB / ID: 4ly9
タイトル
Human GKRP complexed to AMG-1694 [(2R)-1,1,1-trifluoro-2-{4-[(2S)-2-{[(3S)-3-methylmorpholin-4-yl]methyl}-4-(thiophen-2-ylsulfonyl)piperazin-1-yl]phenyl}propan-2-ol] and sorbitol-6-phosphate
要素
Glucokinase regulatory protein
キーワード
Carbohydrate Binding protein / Regulatory protein / disruptor ligand complex / SIS domains / GKRP binds to GK / Liver
機能・相同性
機能・相同性情報
negative regulation of glucokinase activity / glucose sensor activity / carbohydrate derivative metabolic process / fructose-6-phosphate binding / kinase inhibitor activity / urate metabolic process / Regulation of Glucokinase by Glucokinase Regulatory Protein / Defective TPR may confer susceptibility towards thyroid papillary carcinoma (TPC) / response to fructose / enzyme inhibitor activity ...negative regulation of glucokinase activity / glucose sensor activity / carbohydrate derivative metabolic process / fructose-6-phosphate binding / kinase inhibitor activity / urate metabolic process / Regulation of Glucokinase by Glucokinase Regulatory Protein / Defective TPR may confer susceptibility towards thyroid papillary carcinoma (TPC) / response to fructose / enzyme inhibitor activity / triglyceride homeostasis / response to glucose / protein import into nucleus / glucose homeostasis / carbohydrate binding / enzyme binding / mitochondrion / nucleoplasm / cytosol / cytoplasm 類似検索 - 分子機能
: / Glucokinase regulatory protein, second SIS domain / C-terminal lid domain of glucokinase regulatory protein / Glucokinase regulatory protein N-terminal SIS domain / Glucokinase regulatory protein, conserved site / N-acetylmuramic acid 6-phosphate etherase/glucokinase regulatory protein / Glucokinase regulatory protein family signature. / SIS domain / SIS domain profile. / SIS domain superfamily ...: / Glucokinase regulatory protein, second SIS domain / C-terminal lid domain of glucokinase regulatory protein / Glucokinase regulatory protein N-terminal SIS domain / Glucokinase regulatory protein, conserved site / N-acetylmuramic acid 6-phosphate etherase/glucokinase regulatory protein / Glucokinase regulatory protein family signature. / SIS domain / SIS domain profile. / SIS domain superfamily / Glucose-6-phosphate isomerase like protein; domain 1 / Rossmann fold / 3-Layer(aba) Sandwich / Alpha Beta 類似検索 - ドメイン・相同性
Chem-1YY / IODIDE ION / D-SORBITOL-6-PHOSPHATE / Glucokinase regulatory protein 類似検索 - 構成要素