登録情報 | データベース: PDB / ID: 4pxz |
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タイトル | Crystal structure of P2Y12 receptor in complex with 2MeSADP |
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要素 | P2Y purinoceptor 12, Soluble cytochrome b562 |
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キーワード | MEMBRANE PROTEIN / purinergic receptor P2Y12 / agonist-bound / G-protein coupled receptor (GPCR) / signaling protein-agonist complex / PSI-Biology / GPCR Network / Structural Genomics / signaling membrane protein / GPCR / platelet activation / membrane |
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機能・相同性 | 機能・相同性情報
visual system development / positive regulation of integrin activation by cell surface receptor linked signal transduction / cerebral cortex radial glia-guided migration / regulation of microglial cell migration / G protein-coupled ADP receptor activity / P2Y receptors / cell body membrane / G protein-coupled purinergic nucleotide receptor activity / positive regulation of monoatomic ion transport / positive regulation of microglial cell migration ...visual system development / positive regulation of integrin activation by cell surface receptor linked signal transduction / cerebral cortex radial glia-guided migration / regulation of microglial cell migration / G protein-coupled ADP receptor activity / P2Y receptors / cell body membrane / G protein-coupled purinergic nucleotide receptor activity / positive regulation of monoatomic ion transport / positive regulation of microglial cell migration / hemostasis / G protein-coupled adenosine receptor activity / cell projection membrane / regulation of chemotaxis / substrate-dependent cell migration, cell extension / positive regulation of chemotaxis / cell projection organization / positive regulation of ruffle assembly / positive regulation of cell adhesion mediated by integrin / lamellipodium assembly / cellular response to ATP / response to axon injury / monoatomic ion transport / adenylate cyclase-inhibiting G protein-coupled receptor signaling pathway / guanyl-nucleotide exchange factor activity / platelet aggregation / establishment of localization in cell / electron transport chain / calcium-mediated signaling / platelet activation / ADP signalling through P2Y purinoceptor 12 / phospholipase C-activating G protein-coupled receptor signaling pathway / G alpha (i) signalling events / periplasmic space / positive regulation of phosphatidylinositol 3-kinase/protein kinase B signal transduction / electron transfer activity / iron ion binding / G protein-coupled receptor signaling pathway / heme binding / cell surface / membrane / plasma membrane類似検索 - 分子機能 P2Y12 purinoceptor / Cytochrome b562 / Cytochrome b562 / Cytochrome c/b562 / G protein-coupled receptor, rhodopsin-like / GPCR, rhodopsin-like, 7TM / G-protein coupled receptors family 1 profile. / 7 transmembrane receptor (rhodopsin family)類似検索 - ドメイン・相同性 Chem-6AD / CHOLESTEROL / (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate / DI(HYDROXYETHYL)ETHER / Soluble cytochrome b562 / P2Y purinoceptor 12類似検索 - 構成要素 |
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生物種 | Homo sapiens (ヒト) Escherichia coli (大腸菌) |
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手法 | X線回折 / シンクロトロン / 分子置換 / 解像度: 2.5 Å |
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データ登録者 | Zhang, J. / Zhang, K. / Gao, Z.G. / Paoletta, S. / Zhang, D. / Han, G.W. / Li, T. / Ma, L. / Zhang, W. / Muller, C.E. ...Zhang, J. / Zhang, K. / Gao, Z.G. / Paoletta, S. / Zhang, D. / Han, G.W. / Li, T. / Ma, L. / Zhang, W. / Muller, C.E. / Yang, H. / Jiang, H. / Cherezov, V. / Katritch, V. / Jacobson, K.A. / Stevens, R.C. / Wu, B. / Zhao, Q. / GPCR Network (GPCR) |
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引用 | ジャーナル: Nature / 年: 2014 タイトル: Agonist-bound structure of the human P2Y12 receptor 著者: Zhang, J. / Zhang, K. / Gao, Z.G. / Paoletta, S. / Zhang, D. / Han, G.W. / Li, T. / Ma, L. / Zhang, W. / Muller, C.E. / Yang, H. / Jiang, H. / Cherezov, V. / Katritch, V. / Jacobson, K.A. / ...著者: Zhang, J. / Zhang, K. / Gao, Z.G. / Paoletta, S. / Zhang, D. / Han, G.W. / Li, T. / Ma, L. / Zhang, W. / Muller, C.E. / Yang, H. / Jiang, H. / Cherezov, V. / Katritch, V. / Jacobson, K.A. / Stevens, R.C. / Wu, B. / Zhao, Q. |
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履歴 | 登録 | 2014年3月25日 | 登録サイト: RCSB / 処理サイト: PDBJ |
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改定 1.0 | 2014年4月30日 | Provider: repository / タイプ: Initial release |
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改定 1.1 | 2014年5月28日 | Group: Database references |
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改定 1.2 | 2014年9月3日 | Group: Derived calculations |
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改定 1.3 | 2017年8月16日 | Group: Refinement description / Source and taxonomy / カテゴリ: entity_src_gen / software |
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改定 1.4 | 2017年11月22日 | Group: Refinement description / カテゴリ: software / Item: _software.name |
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改定 1.5 | 2023年11月8日 | Group: Data collection / Database references ...Data collection / Database references / Derived calculations / Refinement description カテゴリ: chem_comp_atom / chem_comp_bond ...chem_comp_atom / chem_comp_bond / database_2 / pdbx_initial_refinement_model / struct_ref_seq_dif / struct_site Item: _database_2.pdbx_DOI / _database_2.pdbx_database_accession ..._database_2.pdbx_DOI / _database_2.pdbx_database_accession / _struct_ref_seq_dif.details / _struct_site.pdbx_auth_asym_id / _struct_site.pdbx_auth_comp_id / _struct_site.pdbx_auth_seq_id |
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