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-Structure paper
Title | Mode of action of DNA-competitive small molecule inhibitors of tyrosyl DNA phosphodiesterase 2. |
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Journal, issue, pages | Biochem. J., Vol. 473, Page 1869-1879, Year 2016 |
Publish date | Mar 31, 2016 (structure data deposition date) |
![]() | Hornyak, P. / Askwith, T. / Walker, S. / Komulainen, E. / Paradowski, M. / Pennicott, L.E. / Bartlett, E.J. / Brissett, N.C. / Raoof, A. / Watson, M. ...Hornyak, P. / Askwith, T. / Walker, S. / Komulainen, E. / Paradowski, M. / Pennicott, L.E. / Bartlett, E.J. / Brissett, N.C. / Raoof, A. / Watson, M. / Jordan, A.M. / Ogilvie, D.J. / Ward, S.E. / Atack, J.R. / Pearl, L.H. / Caldecott, K.W. / Oliver, A.W. |
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Methods | X-ray diffraction |
Resolution | 1.7 - 3.4 Å |
Structure data | ![]() PDB-5j3p: ![]() PDB-5j3s: ![]() PDB-5j3z: ![]() PDB-5j42: |
Chemicals | ![]() ChemComp-MG: ![]() ChemComp-GOL: ![]() ChemComp-HOH: ![]() ChemComp-6FQ: ![]() ChemComp-EDO: ![]() ChemComp-ACT: ![]() ChemComp-6FV: ![]() ChemComp-TLA: ![]() ChemComp-MN: |
Source |
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![]() | HYDROLASE / tyrosyl / DNA phosphodiesterase 2 / catalytic domain / tyrosyl DNA phosphodiesterase 2 catalytic domain |