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-Structure paper
Title | Mode of action of DNA-competitive small molecule inhibitors of tyrosyl DNA phosphodiesterase 2. |
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Journal, issue, pages | Biochem. J., Vol. 473, Page 1869-1879, Year 2016 |
Publish date | Mar 31, 2016 (structure data deposition date) |
Authors | Hornyak, P. / Askwith, T. / Walker, S. / Komulainen, E. / Paradowski, M. / Pennicott, L.E. / Bartlett, E.J. / Brissett, N.C. / Raoof, A. / Watson, M. ...Hornyak, P. / Askwith, T. / Walker, S. / Komulainen, E. / Paradowski, M. / Pennicott, L.E. / Bartlett, E.J. / Brissett, N.C. / Raoof, A. / Watson, M. / Jordan, A.M. / Ogilvie, D.J. / Ward, S.E. / Atack, J.R. / Pearl, L.H. / Caldecott, K.W. / Oliver, A.W. |
External links | Biochem. J. / PubMed:27099339 |
Methods | X-ray diffraction |
Resolution | 1.7 - 3.4 Å |
Structure data | PDB-5j3p: PDB-5j3s: PDB-5j3z: PDB-5j42: |
Chemicals | ChemComp-MG: ChemComp-GOL: ChemComp-HOH: ChemComp-6FQ: ChemComp-EDO: ChemComp-ACT: ChemComp-6FV: ChemComp-TLA: ChemComp-MN: |
Source |
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Keywords | HYDROLASE / tyrosyl / DNA phosphodiesterase 2 / catalytic domain / tyrosyl DNA phosphodiesterase 2 catalytic domain |