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-Structure paper
タイトル | Structure-guided optimization of protein kinase inhibitors reverses aminoglycoside antibiotic resistance. |
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ジャーナル・号・ページ | Biochem. J., Vol. 454, Page 191-200, Year 2013 |
掲載日 | 2012年4月6日 (構造データの登録日) |
著者 | Stogios, P.J. / Spanogiannopoulos, P. / Evdokimova, E. / Egorova, O. / Shakya, T. / Todorovic, N. / Capretta, A. / Wright, G.D. / Savchenko, A. |
リンク | Biochem. J. / PubMed:23758273 |
手法 | X線回折 |
解像度 | 1.863 - 2.71 Å |
構造データ | PDB-4ej7: PDB-4feu: PDB-4fev: PDB-4few: PDB-4fex: PDB-4gkh: PDB-4gki: |
化合物 | ChemComp-ATP: ChemComp-CA: ChemComp-PEG: ChemComp-HOH: ChemComp-KAN: ChemComp-537: ChemComp-ACT: ChemComp-PP1: ChemComp-NA: ChemComp-PP2: ChemComp-CL: ChemComp-0TO: ChemComp-0J9: ChemComp-0JN: |
由来 |
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キーワード | TRANSFERASE / CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES / CSGID / NIAID / National Institute of Allergy and Infectious Diseases / EUKARYOTIC PROTEIN KINASE-LIKE FOLD / ALPHA/BETA PROTEIN / PHOSPHOTRANSFERASE / AMINOGLYCOSIDE PHOSPHOTRANSFERASE / ANTIBIOTIC RESISTANCE / AMINOGLYCOSIDES / KANAMYCIN / GTP / INTRACELLULAR / TRANSFERASE/TRANSFERASE INHIBITOR / anthrapyrazolone / SP600125 / protein kinase inhibitor / TRANSFERASE-TRANSFERASE INHIBITOR complex / pyrazolopyrimidine / PP1 / PP2 / tyrphostin / 4-anilinoquinazoline / tyrphostin AG1478 / AG1478 / 1-NA-PP1 / BUMPED KINASE INHIBITOR / BKI / 1-NM-PP1 |