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-Structure paper
タイトル | Design of potent selective zinc-mediated serine protease inhibitors. |
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ジャーナル・号・ページ | Nature, Vol. 391, Page 608-612, Year 1998 |
掲載日 | 1999年7月21日 (構造データの登録日) |
![]() | Katz, B.A. / Clark, J.M. / Finer-Moore, J.S. / Jenkins, T.E. / Johnson, C.R. / Ross, M.J. / Luong, C. / Moore, W.R. / Stroud, R.M. |
![]() | ![]() ![]() |
手法 | X線回折 |
解像度 | 1.37 - 2.2 Å |
構造データ | ![]() PDB-1c1n: ![]() PDB-1c1o: ![]() PDB-1c1p: ![]() PDB-1c1q: ![]() PDB-1c1r: ![]() PDB-1c1t: ![]() PDB-1c1u: ![]() PDB-1c1v: ![]() PDB-1c1w: ![]() PDB-1c2d: ![]() PDB-1c2e: ![]() PDB-1c2f: ![]() PDB-1c2g: ![]() PDB-1c2h: ![]() PDB-1c2i: ![]() PDB-1c2j: ![]() PDB-1c2k: ![]() PDB-1c2l: ![]() PDB-1c2m: ![]() PDB-1xuf: ![]() PDB-1xug: ![]() PDB-1xuh: ![]() PDB-1xui: ![]() PDB-1xuj: ![]() PDB-1xuk: |
化合物 | ![]() ChemComp-CA: ![]() ChemComp-ZN: ![]() ChemComp-SO4: ![]() ChemComp-BEN: ![]() ChemComp-HOH: ![]() ChemComp-MG: ![]() ChemComp-BAI: ![]() ChemComp-DMS: ![]() ChemComp-BAB: ![]() ChemComp-NA: ![]() ChemComp-BAH: ![]() ChemComp-BAK: ![]() ChemComp-CL: ![]() ChemComp-ABI: ![]() ChemComp-BAZ: ![]() ChemComp-CO: ![]() ChemComp-BAO: ![]() ChemComp-BOZ: |
由来 |
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![]() | HYDROLASE/HYDROLASE INHIBITOR / ZN(II)-MEDIATED SERINE PROTEASE INHIBITORS / PH DEPENDENCE / ZN(II) AFFINITY STUCTURE-BASED DRUG DESIGN / SERINE PROTEASE / HYDROLASE-HYDROLASE INHIBITOR COMPLEX / SERINE PROTEASE SERINE PROTEASE/INHIBITOR / SERINE PROTEASE/INHIBITOR / BLOOD CLOTTING/HYDROLASE INHIBITOR / BLOOD CLOTTING-HYDROLASE INHIBITOR COMPLEX / BLOOD CLOTTING / COMPLEX / TRYPSIN-ZN+2-SMALL MOLECULE LIGAND / DESIGNED SMALL MOLECULE LIGAND WITH NANOMOLAR AFFINITY / TRYPSIN-COBALT-SMALL MOLECULE LIGAND / DESIGNED SMALL MOLECULE LIGAND WITH MICROMOLAR AFFINITY / TRYPSIN-SMALL MOLECULE LIGAND / TRYPSIN-SULFATE-SMALL MOLECULE LIGAND |