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3W1F
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BU of 3w1f by Molmil
Crystal structure of Human MPS1 catalytic domain in complex with 5-(5-ethoxy-6-(1-methyl-1H-pyrazol-4-yl)-1H-indazol-3-yl)-2-methylbenzenesulfonamide
Descriptor: 5-[5-ethoxy-6-(1-methyl-1H-pyrazol-4-yl)-1H-indazol-3-yl]-2-methylbenzenesulfonamide, Dual specificity protein kinase TTK
Authors:Kusakabe, K, Ide, N, Daigo, Y, Tachibana, Y, Itoh, T, Yamamoto, T, Hashizume, H, Hato, Y, Higashino, K, Okano, Y, Sato, Y, Inoue, M, Iguchi, M, Kanazawa, T, Ishioka, Y, Dohi, K, Kido, Y, Sakamoto, S, Yasuo, K, Maeda, M, Higaki, M, Ueda, K, Yoshizawa, H, Baba, Y, Shiota, T, Murai, H, Nakamura, Y.
Deposit date:2012-11-14
Release date:2013-06-26
Last modified:2024-03-20
Method:X-RAY DIFFRACTION (2.7 Å)
Cite:Indazole-based potent and cell-active Mps1 kinase inhibitors: rational design from pan-kinase inhibitor anthrapyrazolone (SP600125)
J.Med.Chem., 56, 2013
3OB9
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BU of 3ob9 by Molmil
Structure of the human MSL3 chromo-barrel domain at 2.5 Angstrom resolution
Descriptor: 2-[N-CYCLOHEXYLAMINO]ETHANE SULFONIC ACID, Male-specific lethal 3-like 1 (Drosophila), isoform CRA_c, ...
Authors:Moore, S.A, Ferhatoglu, Y.
Deposit date:2010-08-06
Release date:2010-10-13
Last modified:2023-09-06
Method:X-RAY DIFFRACTION (2.5 Å)
Cite:Structure of the human MSL3 chromo-barrel domain at 2.5 Angstrom resolution
J.Biol.Chem., 2010
7DC0
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BU of 7dc0 by Molmil
Crystal structure of glycan-free Pseudomonas taiwanensis lectin
Descriptor: Lectin, SULFATE ION
Authors:Oda, K, Matoba, Y.
Deposit date:2020-10-23
Release date:2021-04-28
Last modified:2023-11-29
Method:X-RAY DIFFRACTION (1.88 Å)
Cite:Lectins engineered to favor a glycan-binding conformation have enhanced antiviral activity.
J.Biol.Chem., 296, 2021
7DC4
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BU of 7dc4 by Molmil
Crystal structure of glycan-bound Pseudomonas taiwanensis lectin
Descriptor: Lectin, SULFATE ION, alpha-D-mannopyranose-(1-3)-[alpha-D-mannopyranose-(1-6)]alpha-D-mannopyranose-(1-6)-[alpha-D-mannopyranose-(1-3)]beta-D-mannopyranose
Authors:Oda, K, Matoba, Y.
Deposit date:2020-10-23
Release date:2021-04-28
Last modified:2023-11-29
Method:X-RAY DIFFRACTION (0.95 Å)
Cite:Lectins engineered to favor a glycan-binding conformation have enhanced antiviral activity.
J.Biol.Chem., 296, 2021

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