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PDB: 1 results

4BJX
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BU of 4bjx by Molmil
N-TERMINAL BROMODOMAIN OF HUMAN BRD4 WITH GSK1324726A (I-BET726)
Descriptor: 4-[(2S,4R)-1-acetyl-4-[(4-chlorophenyl)amino]-2-methyl-1,2,3,4-tetrahydroquinolin-6-yl]benzoic acid, BROMODOMAIN-CONTAINING PROTEIN 4
Authors:Chung, C.
Deposit date:2013-04-20
Release date:2013-10-02
Last modified:2019-05-15
Method:X-RAY DIFFRACTION (1.59 Å)
Cite:Bet Inhibition Silences Expression of Mycn and Bcl2 and Induces Cytotoxicity in Neuroblastoma Tumor Models.
Plos One, 8, 2013

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